Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 1349
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11014((-)-(S)1 | (5S)-5-(4-chlorophenyl)-3-(4-methylphen...)
Affinity DataKi:  1nM ΔG°:  -53.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11004(5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  1.5nM ΔG°:  -52.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11015((5R)-5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dih...)
Affinity DataKi:  2.70nM ΔG°:  -51.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11006(5-(furan-2-yl)-3-(4-methylphenyl)-4,5-dihydro-1H-p...)
Affinity DataKi:  4nM ΔG°:  -50.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11016((5S)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  5nM ΔG°:  -49.4kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11005(3,5-bis(4-methylphenyl)-4,5-dihydro-1H-pyrazole-1-...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11007(5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dihydro-...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11010(5-(4-chlorophenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  6nM ΔG°:  -49.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11008(3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  7nM ΔG°:  -48.6kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11009(3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydro-1H-p...)
Affinity DataKi:  8nM ΔG°:  -48.2kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11005(3,5-bis(4-methylphenyl)-4,5-dihydro-1H-pyrazole-1-...)
Affinity DataKi:  10nM ΔG°:  -47.7kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11011(5-(4-methylphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  10nM ΔG°:  -47.7kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11017((5R)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  12nM ΔG°:  -47.2kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11015((5R)-5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dih...)
Affinity DataKi:  13nM ΔG°:  -47.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11012(5-(furan-2-yl)-3-(thiophen-2-yl)-4,5-dihydro-1H-py...)
Affinity DataKi:  20nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11013(3,5-bis(thiophen-2-yl)-4,5-dihydro-1H-pyrazole-1-c...)
Affinity DataKi:  27nM ΔG°:  -45.1kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11004(5-(4-chlorophenyl)-3-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  31nM ΔG°:  -44.7kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11010(5-(4-chlorophenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  41nM ΔG°:  -44.0kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11008(3-(4-fluorophenyl)-5-(4-methylphenyl)-4,5-dihydro-...)
Affinity DataKi:  50nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11011(5-(4-methylphenyl)-3-(thiophen-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  50nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11013(3,5-bis(thiophen-2-yl)-4,5-dihydro-1H-pyrazole-1-c...)
Affinity DataKi:  50nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11012(5-(furan-2-yl)-3-(thiophen-2-yl)-4,5-dihydro-1H-py...)
Affinity DataKi:  50nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Bovine)
Sapienza University of Rome

LigandPNGBDBM11014((-)-(S)1 | (5S)-5-(4-chlorophenyl)-3-(4-methylphen...)
Affinity DataKi:  50nM ΔG°:  -43.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11006(5-(furan-2-yl)-3-(4-methylphenyl)-4,5-dihydro-1H-p...)
Affinity DataKi:  170nM ΔG°:  -40.3kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11009(3-(4-fluorophenyl)-5-(furan-2-yl)-4,5-dihydro-1H-p...)
Affinity DataKi:  370nM ΔG°:  -38.3kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11007(5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dihydro-...)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.7kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11017((5R)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  1.40E+3nM ΔG°:  -34.9kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Bovine)
Sapienza University of Rome

LigandPNGBDBM11016((5S)-5-(4-chlorophenyl)-3-(4-fluorophenyl)-4,5-dih...)
Affinity DataKi:  2.40E+3nM ΔG°:  -33.5kJ/molepH: 7.4 T: 2°CAssay Description:MAO A and MAO B activities were determined spectrophotometrically using kynuramine as substrates. Fluorimetric measurements were recorded with a Perk...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/12/2006
Entry Details Article
PubMed