Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50017104
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177501({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148292(1-(PHENYLMETHYL)CYCLOPENTYL[(1S)-1-FORMYLPENTYL]CA...)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148298(((S)-1-Formyl-pentyl)-carbamic acid (R)-1-benzyl-2...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177494({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 0.940nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177503({(S)-1-[(2,3-dihydro-indole-1-carbonyl)-hydrazonom...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148296((S)-1-phenylpropan-2-yl (S)-1-oxohexan-2-ylcarbama...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177501({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148298(((S)-1-Formyl-pentyl)-carbamic acid (R)-1-benzyl-2...)
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148298(((S)-1-Formyl-pentyl)-carbamic acid (R)-1-benzyl-2...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human cathepsin H in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177501({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human cathepsin B in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177512({(S)-1-[(2,2,2-trifluoro-acetyl)-hydrazonomethyl]-...)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148298(((S)-1-Formyl-pentyl)-carbamic acid (R)-1-benzyl-2...)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human cathepsin B in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50137822(CHEMBL204666 | CHEMBL96823 | ((S)-1-Formyl-3-methy...)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177491({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177489({(S)-1-[(pyrrolidine-1-carbonyl)-hydrazonomethyl]-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148296((S)-1-phenylpropan-2-yl (S)-1-oxohexan-2-ylcarbama...)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human cathepsin H in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177511(tert-butyl N-[(1E,2S)-1-{[(diethylcarbamoyl)amino]...)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177517(tert-butyl N-[(1E,2S)-1-({[methyl(2-phenylethyl)ca...)
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177495({(S)-1-[(2,3-dihydro-indole-1-carbonyl)-hydrazonom...)
Affinity DataIC50: 48nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50137790([(S)-1-(4-Bromo-1H-pyrazol-3-ylaminooxalyl)-pentyl...)
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177496({(S)-1-[(piperidine-1-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 58nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177506({(S)-1-[(3,4-dihydro-2H-quinoline-1-carbonyl)-hydr...)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177513(tert-butyl (1S)-1-({[(dimethylamino)carbonyl]hydra...)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177521(tert-butyl (1S)-1-({[(dimethylamino)sulfonyl]hydra...)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177502({(S)-1-[(3,4-dihydro-1H-isoquinoline-2-carbonyl)-h...)
Affinity DataIC50: 93nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177509({(S)-3-methyl-1-[(morpholine-4-carbonyl)-hydrazono...)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177494({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 130nMAssay Description:Inhibition of rat cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177516(N'-[(S)-2-tert-butoxycarbonylamino-hexylidene]-hyd...)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177497(tert-butyl N-[(1E,2S)-1-{[(tert-butylcarbamoyl)ami...)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177488(tert-butyl N-[(1E,2S)-1-({[(propan-2-yl)carbamoyl]...)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177514(tert-butyl N-[(1E,2S)-1-{[N-(propan-2-yl)-(C-sulfa...)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177492(methyl (2-{(2S)-2-[(tert-butoxycarbonyl)amino]hexy...)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177501({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human cathepsin H in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177508({(S)-1-[(3-methyl-butyryl)-hydrazonomethyl]-pentyl...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177520([(S)-1-(benzoyl-hydrazonomethyl)-pentyl]-carbamic ...)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPro-cathepsin H(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177494({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human cathepsin H in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177493(tert-butyl N-[(1E,2S)-1-({[(2-phenylethyl)carbamoy...)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177494({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human cathepsin B in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177523(tert-butyl (1S)-1-({[(methylamino)carbonyl]hydrazo...)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177498(tert-butyl (1S)-1-{[(aminocarbonyl)hydrazono]methy...)
Affinity DataIC50: 350nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177510(tert-butyl N-[(1E,2S)-1-{[(phenylcarbamoyl)amino]i...)
Affinity DataIC50: 400nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177505(tert-butyl N-[(1E,2S)-1-{[(benzylcarbamoyl)amino]i...)
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin B(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148296((S)-1-phenylpropan-2-yl (S)-1-oxohexan-2-ylcarbama...)
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant human cathepsin B in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177522({(S)-1-[(4,5-dihydro-thiazol-3-yl)-hydrazonomethyl...)
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177499(ethyl 3-({N'-[(1E,2S)-2-{[(tert-butoxy)carbonyl]am...)
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177500(tert-butyl (1S)-1-({[(ethylamino)carbonyl]hydrazon...)
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177507(ethyl 2-({N'-[(1E,2S)-2-{[(tert-butoxy)carbonyl]am...)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCathepsin K(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177519(tert-butyl N-[(1E,2S)-1-({methyl[methyl(2-phenylet...)
Affinity DataIC50: 520nMAssay Description:Inhibition of recombinant human cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50177494({(S)-1-[(morpholine-4-carbonyl)-hydrazonomethyl]-p...)
Affinity DataIC50: 540nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50148296((S)-1-phenylpropan-2-yl (S)-1-oxohexan-2-ylcarbama...)
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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