Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50017106
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177543(1-(3-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177530(4-((1H-imidazol-4-yl)methyl)-1-(3-(3-(cyclohexylox...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177531(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177536(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177538(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175839(4-((1H-imidazol-4-yl)methyl)-1-(3-phenoxypropyl)pi...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177551(4-((1H-imidazol-4-yl)methyl)-N-(thiazol-2-yl)piper...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177535(N-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177542(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177544(1-(4-(2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177532(4-((1H-imidazol-4-yl)methyl)-1-(3-(4-(cyclohexylox...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177546(4-((1H-imidazol-4-yl)methyl)-N-(pyrimidin-2-yl)pip...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177556(5-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177541(5-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177528(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177548(3-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177550(5-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177529(3-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177527(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177555(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177534(1-(4-(4-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177549(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177552(3-(4-((4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177526((4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177533((6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177545((4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50175839(4-((1H-imidazol-4-yl)methyl)-1-(3-phenoxypropyl)pi...)
Affinity DataIC50: 30nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177547(N,N-dimethyl-3-(4-(piperidin-1-ylmethyl)phenoxy)pr...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177539(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177540(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-N-(...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177524(2-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177554(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177553(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177537(6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177532(4-((1H-imidazol-4-yl)methyl)-1-(3-(4-(cyclohexylox...)
Affinity DataIC50: 300nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177548(3-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataIC50: 300nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetHistamine H3 receptor(Guinea pig)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177525(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(...)
Affinity DataKi:  315nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from guinea pig histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177527(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataIC50: 900nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177531(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CYP2D6 by supersome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177555(1-(4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177525(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177537(6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177533((6-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177530(4-((1H-imidazol-4-yl)methyl)-1-(3-(3-(cyclohexylox...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177551(4-((1H-imidazol-4-yl)methyl)-N-(thiazol-2-yl)piper...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177545((4-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CYP2D6 by supersome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177543(1-(3-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177541(5-(3-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)p...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177554(1-(4-((1H-imidazol-4-yl)methyl)piperidin-1-yl)-3-(...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50177544(1-(4-(2-(4-((1H-imidazol-4-yl)methyl)piperidin-1-y...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of CYP2D6 by human liver microsome assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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