Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50017209
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179064(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179070(8-aminomethyl-1,2,3,5,6,11-hexahydro-5,11-diaza-be...)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179068(8-bromo-1,2,3,5,6,11-hexahydro-5,11-diaza-benzo[a]...)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177482(4,5,6,7-tetrahydro-1Hcyclopenta[a]pyrrolo[3,4-c]ca...)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177476(1,2,3,5,6,11-hexahydro-5,11-diaza-benzo[a]trinden-...)
Affinity DataIC50: 56nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179057(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179056(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179061(2,6-diamino-hexanoic acid (4-oxo-2,3,4,5,6,11-hexa...)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179062(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179069(8-(morpholine-4-carbonyl)-1,2,3,5,6,11-hexahydro-5...)
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179060(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 105nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179059(8-chloro-1,2,3,5,6,11-hexahydro-5,11-diaza-benzo[a...)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179063(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 161nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179058(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179067(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 165nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179054(8-methyl-1,2,3,5,6,11-hexahydro-5,11-diaza-benzo[a...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179055(4-oxo-2,3,4,5,6,11-hexahydro-1H-5,11-diaza-benzo[a...)
Affinity DataIC50: 237nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179071({5-tert-butoxycarbonylamino-5-[(4-oxo-2,3,4,5,6,11...)
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179065(11-methyl-1,2,3,5,6,11-hexahydro-5,11-diaza-benzo[...)
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179072(4-oxo-1,2,3,4,6,11-hexahydro-5,11-diaza-benzo[a]tr...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50177479(1,2,3,4,5,11-hexahydro-5,11-diaza-benzo[a]trinden-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPoly [ADP-ribose] polymerase 1(Human)
Cephalon

Curated by ChEMBL
LigandPNGBDBM50179066(5,11-dimethyl-1,2,3,5,6,11-hexahydro-5,11-diaza-be...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human PARP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed