Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50017228
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  2nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  10nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  14nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  18nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  80nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  80nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 92nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 105nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  125nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataIC50: 127nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataIC50: 152nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179242(2-{4-[3-(3-phenyl-7-propylbenzo[b]furan-6-yloxy)pr...)
Affinity DataEC50:  169nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179237(2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  186nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  220nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179236(2-(5-(3-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  230nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  243nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  280nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179229(2-{5-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  290nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  311nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  320nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179231({5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazol-...)
Affinity DataEC50:  370nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179228(2-{5-[3-(7-propyl-1H-indol-6-yl)propoxy]indol-1-yl...)
Affinity DataEC50:  420nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataIC50: 422nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179225(2-{4-[3-(3-phenyl-7-propylbenzo[d]isoxazol-6-yloxy...)
Affinity DataEC50:  430nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179231({5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazol-...)
Affinity DataEC50:  474nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataEC50:  500nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179240(3-{5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 584nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179237(2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  610nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179227(2-(5-(2-(7-propyl-3-(trifluoromethyl)benzo[d]isoxa...)
Affinity DataEC50:  690nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179226(2-{5-[3-(3-cyano-7-propyl-1H-indol-6-yloxy)propoxy...)
Affinity DataIC50: 759nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179233(2-{4-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 774nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179231({5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazol-...)
Affinity DataEC50:  898nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179235(2-{5-[4-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.04E+3nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 1.05E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179243(2-{5-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 1.05E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179248(3-{4-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179231({5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazol-...)
Affinity DataIC50: 1.12E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179240(3-{5-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.20E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179228(2-{5-[3-(7-propyl-1H-indol-6-yl)propoxy]indol-1-yl...)
Affinity DataEC50:  1.21E+3nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179249(2-ethyl-2-{4-[3-(7-propyl-3-trifluoromethylbenzo[d...)
Affinity DataIC50: 1.28E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179238(2-{4-[2-methyl-3-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179234(2-{6-[3-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.35E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179244(2-{5-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50: 1.37E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179239(2-{4-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50: 1.45E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179243(2-{5-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataEC50:  1.49E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179241(2-{4-[2-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataIC50: 1.68E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179230(2-ethyl-2-{5-[3-(7-propyl-3-trifluoromethylbenzo[d...)
Affinity DataIC50: 1.71E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179247(2-{4-[5-(7-propyl-3-trifluoromethylbenzo[d]isoxazo...)
Affinity DataIC50: 1.78E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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