Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50037678
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179532(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 2.70nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179555((S)-2-(biphenyl-3-ylamino)-4-methyl-pentanoic acid...)
Affinity DataIC50: 3.80nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179548(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 3.90nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179543((4-{(S)-2-[(S)-2-(biphenyl-3-ylamino)-4-methyl-pen...)
Affinity DataIC50: 4.5nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179547([4-((S)-2-{[1-(biphenyl-3-ylamino)-cyclohexanecarb...)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179539([4-((S)-2-{[1-(biphenyl-3-ylamino)-cyclohexanecarb...)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179542(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 5.60nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179558((4-{(S)-2-[(S)-2-(biphenyl-3-ylamino)-4-methyl-pen...)
Affinity DataIC50: 6.40nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179551(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179559((S)-2-(biphenyl-3-ylamino)-4-methyl-pentanoic acid...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179538((S)-2-(biphenyl-3-ylamino)-4-methyl-pentanoic acid...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179549((S)-2-(biphenyl-3-ylamino)-4-methyl-pentanoic acid...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179556((S)-2-(3-cyclohexylphenylamino)-N-(2-(4-methoxyphe...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179560(N-(2-(4-methoxyphenylamino)ethyl)-4-methyl-2-(3-ph...)
Affinity DataIC50: 69nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179550(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 82nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179534(1-(biphenyl-3-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 83nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179537(2-(biphenyl-3-yloxy)-4-methyl-pentanoic acid [2-(4...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50113676({1-[2-(4-Methoxy-phenylamino)-ethylcarbamoyl]-3-me...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179553(1-(4-cyclohexylphenoxy)-N-(2-(4-methoxyphenylamino...)
Affinity DataIC50: 99nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179561(2-(biphenyl-4-yloxy)-4-methyl-pentanoic acid [2-(4...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179540(1-(biphenyl-4-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179557(1-(4-ethylphenoxy)-N-(2-(4-methoxyphenylamino)ethy...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179546(1-(biphenyl-4-yloxy)-cyclohexanecarboxylic acid [2...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179536(1-(4-isopropylphenoxy)-N-(2-(4-methoxyphenylamino)...)
Affinity DataIC50: 200nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179541(1-(biphenyl-3-yloxy)-cyclohexanecarboxylic acid [2...)
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179545(N-(2-(4-methoxyphenylamino)ethyl)-4-methyl-2-(4-ph...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179533(2-(biphenyl-2-yloxy)-4-methyl-pentanoic acid [2-(4...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179535(N-(2-(4-methoxyphenylamino)ethyl)-4-methyl-2-pheno...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179554(N-(2-(4-methoxyphenylamino)ethyl)-1-phenoxycyclohe...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179552(N-(2-(4-methoxyphenylamino)ethyl)-1-(phenylamino)c...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed
TargetCathepsin K(Human)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50179544(1-(biphenyl-2-ylamino)-cyclohexanecarboxylic acid ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against recombinant human Cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/6/2012
Entry Details Article
PubMed