Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50041442
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184908(cypate-[(RGD)4-NH2]1 | CHEMBL402661)
Affinity DataIC50: 25.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184904(cyclo(RGDfV) (control) | CHEMBL206344)
Affinity DataIC50: 28.7nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184902(cyclo[RGDfK(cypate)] | CHEMBL407126)
Affinity DataIC50: 63.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184906(cypate-[(RGD)4-NH2]2 | CHEMBL429568)
Affinity DataIC50: 79.6nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184903(cypate-[(RGD)2-NH2]2 | CHEMBL415188)
Affinity DataIC50: 104nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184905(cypate-[(RGD)3-NH2]2 | CHEMBL413898)
Affinity DataIC50: 132nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184907(cypate-[(RGD)3-NH2]1 | CHEMBL412767)
Affinity DataIC50: 481nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetIntegrin alpha-V/beta-3(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50184909(cypate-[(RGD)2-NH2]1 | CHEMBL438186)
Affinity DataIC50: 730nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed