Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50017648
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(N-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataEC50:  260nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(N-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataEC50:  400nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  890nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(N-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataEC50:  600nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(N-oleoyl-O-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataEC50:  320nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataEC50:  490nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(N-arachidonoyl-O-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataEC50:  250nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  70nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(N-arachidonoyl-O-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  81nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  180nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185034(N-arachidonoyl-O-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  470nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(N-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185037(O-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185037(O-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(N-oleoyl-O-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185035(N-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataKi:  3.90E+3nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(N-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataKi:  5.40E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185030(O-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL3...)
Affinity DataKi:  8.60E+3nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185029(O-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185029(O-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(N-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185032(N-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185031(N-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185030(O-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL3...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185033(N-oleoyl-O-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185036(N-palmitoyl-O-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50185036(N-palmitoyl-O-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB1 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to human recombinant CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed