Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50017692
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataKi:  0.0500nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185367(H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 | CHEMBL413871)
Affinity DataKi:  3.90nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  4.10nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185365(Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436493 | CH...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185369(H-[Trp-Arg-Nva-Arg-Tyr]2-NH2 | CHEMBL408891)
Affinity DataKi:  5.30nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataKi:  7.5nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50049744([Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2 | NPY-analogs | CHE...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]hPP from human NPY4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185367(H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 | CHEMBL413871)
Affinity DataKi:  30nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185367(H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 | CHEMBL413871)
Affinity DataKi:  50nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]NPY from human NPY1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]NPY from human NPY1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  140nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]NPY from human NPY1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185365(Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436493 | CH...)
Affinity DataKi:  140nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185369(H-[Trp-Arg-Nva-Arg-Tyr]2-NH2 | CHEMBL408891)
Affinity DataKi:  220nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185367(H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 | CHEMBL413871)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  260nMAssay Description:Displacement of [125I]NPY from human NPY2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185368(Pim[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL439884 | CH...)
Affinity DataKi:  260nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185369(H-[Trp-Arg-Nva-Arg-Tyr]2-NH2 | CHEMBL408891)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50049744([Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2 | NPY-analogs | CHE...)
Affinity DataKi:  340nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185365(Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436493 | CH...)
Affinity DataKi:  360nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  390nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185365(Adp[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436493 | CH...)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]NPY from human NPY2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50049744([Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2 | NPY-analogs | CHE...)
Affinity DataEC50:  570nMAssay Description:Agonist activity at human NPY4 receptor in HEK293 cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185364(Sub[-Tyr-Arg-Leu-Arg-Tyr-NH2]2 | CHEMBL415187 | CH...)
Affinity DataKi:  890nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185369(H-[Trp-Arg-Nva-Arg-Tyr]2-NH2 | CHEMBL408891)
Affinity DataKi:  1.05E+3nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185367(H-[Trp-Arg-Nva-Arg-Tyr]3-NH2 | CHEMBL413871)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50185366(Sub[-Trp-Arg-Nva-Arg-Tyr-NH2]2 | CHEMBL436499 | CH...)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at human NPY1 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
University of Cincinnati

Curated by ChEMBL
LigandPNGBDBM50049744([Cys-Trp-Arg-Nva-Arg-Tyr-NH2]2 | NPY-analogs | CHE...)
Affinity DataKi: >3.00E+3nMAssay Description:Agonist activity at human NPY2 receptor in CHO cells by inhibition of forskolin-stimulated cAMP synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed