Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50037706
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50185420(2-(4-{1-[4-(1-carboxy-propoxy)-3-methyl-phenyl]-cy...)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human recombinant PPARalpha by transactivation of TK-MH100x4-LUC reporter gene in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50185421(2-(4-(3-(4-((3-(2,6-dichlorophenyl)-5-isopropyliso...)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human recombinant FXR by transactivation of TK-MH100x4-LUC reporter gene in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM28700(alpha-1081 | procetofenic acid | Fenofibrate | CHE...)
Affinity DataEC50:  9.20E+3nMAssay Description:Agonist activity at human recombinant PPARalpha by transactivation of TK-MH100x4-LUC reporter gene in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBile acid receptor(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM21674(Chenodeoxycholic Acid | CDCA | (4R)-4-[(1S,2S,5R,7...)
Affinity DataEC50:  1.17E+4nMAssay Description:Agonist activity at human recombinant FXR by transactivation of TK-MH100x4-LUC reporter gene in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)