Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50017862
TargetAdenosine receptor A3(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(N-(4-methoxy-phenyl)-2-cyclopentyl-1H-imidazo[4,5-...)
Affinity DataKi:  410nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596(CHEMBL442333 | N-phenyl-2-cyclopentyl-1H-imidazo[4...)
Affinity DataKi:  786nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(N-(4-methyl-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi:  1.19E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(N-(4-chloro-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596(CHEMBL442333 | N-phenyl-2-cyclopentyl-1H-imidazo[4...)
Affinity DataKi:  3.15E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596(CHEMBL442333 | N-phenyl-2-cyclopentyl-1H-imidazo[4...)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(N-(4-methyl-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi:  3.85E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(N-(4-methoxy-phenyl)-2-cyclopentyl-1H-imidazo[4,5-...)
Affinity DataKi:  4.17E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi:  4.69E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187670(N-(4-methyl-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi:  5.22E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187669(N-(4-methoxy-phenyl)-2-cyclopentyl-1H-imidazo[4,5-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(N-(4-chloro-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187671(N-(4-chloro-phenyl)-2-cyclopentyl-1H-imidazo[4,5-c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50187672(CHEMBL207209 | N-(3,4-dichloro-phenyl)-2-cyclopent...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed