Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50018001
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189815(6-amino-4-benzamido-1,2-dihydro-2-(4-methoxyphenyl...)
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity against Cl-IB-MECA inhibited cAMP level in CHO cells transfected with human A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189818(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]tri...)
Affinity DataIC50: 28.3nMAssay Description:Antagonist activity against Cl-IB-MECA inhibited cAMP level in CHO cells transfected with human A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189812(N-benzoyl-N-[2-(4-methoxy-phenyl)-1-oxo-1,2-dihydr...)
Affinity DataIC50: 31.8nMAssay Description:Antagonist activity against Cl-IB-MECA inhibited cAMP level in CHO cells transfected with human A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189805(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]tr...)
Affinity DataIC50: 215nMAssay Description:Antagonist activity against Cl-IB-MECA inhibited cAMP level in CHO cells transfected with human A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189815(6-amino-4-benzamido-1,2-dihydro-2-(4-methoxyphenyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of NECA-stimulated cAMP level in CHO cells transfected with human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189805(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]tr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of NECA-stimulated cAMP level in CHO cells transfected with human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189818(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]tri...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of NECA-stimulated cAMP level in CHO cells transfected with human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189812(N-benzoyl-N-[2-(4-methoxy-phenyl)-1-oxo-1,2-dihydr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of NECA-stimulated cAMP level in CHO cells transfected with human adenosine A2B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189814(N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189810(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  0.810nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189809(N-(6-amino-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189815(6-amino-4-benzamido-1,2-dihydro-2-(4-methoxyphenyl...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50086159(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  1.47nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189817(6-amino-1,2-dihydro-2-phenyl-4-diphenylacetamido-1...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50086146(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189803(6-amino-1,2-dihydro-2-(methoxyphenyl)-4-diphenylac...)
Affinity DataKi:  2.58nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189807(4-benzamido-2-(4-methoxyphenyl)-1,2-dihydro-1,2,4-...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189812(N-benzoyl-N-[2-(4-methoxy-phenyl)-1-oxo-1,2-dihydr...)
Affinity DataKi:  3.29nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189806(N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50086146(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189818(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]tri...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189811(N-(6-amino-2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189820(N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189805(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]tr...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189817(6-amino-1,2-dihydro-2-phenyl-4-diphenylacetamido-1...)
Affinity DataKi:  8.65nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189810(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  10.2nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189806(N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189810(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  18.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189819(6-amino-4-benzamido-1,2-dihydro-2-phenyl-1,2,4-tri...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189813(4-benzamido-6-nitro-2-phenyl-1,2-dihydro-1,2,4-tri...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189818(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]tri...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189808(4-acetamido-2-(4-methoxyphenyl)-1,2-dihydro-1,2,4-...)
Affinity DataKi:  35.7nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189819(6-amino-4-benzamido-1,2-dihydro-2-phenyl-1,2,4-tri...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189805(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro-[1,2,4]tr...)
Affinity DataKi:  44nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189809(N-(6-amino-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  48nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189803(6-amino-1,2-dihydro-2-(methoxyphenyl)-4-diphenylac...)
Affinity DataKi:  77.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189802(N-(6-amino-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50086159(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  87.8nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50086159(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  88.2nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50086159(N-(1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triazolo[4,3-...)
Affinity DataKi:  89.6nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189819(6-amino-4-benzamido-1,2-dihydro-2-phenyl-1,2,4-tri...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189804(4-benzamido-1,2-dihydro-2-(4-nitrophenyl)-1,2,4-tr...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189812(N-benzoyl-N-[2-(4-methoxy-phenyl)-1-oxo-1,2-dihydr...)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50189816(N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[...)
Affinity DataKi:  217nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189808(4-acetamido-2-(4-methoxyphenyl)-1,2-dihydro-1,2,4-...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Università

Curated by ChEMBL
LigandPNGBDBM50189814(N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Università

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]CGS 21680 from adenosine A2A receptor in bovine striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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