Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50035980
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 24nMAssay Description:Compound was tested in vitro for binding affinity towards Dopamine receptor D2 in rat striatal membrane by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 138nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 138nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 203nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50001955(APOKYN | CHEMBL53 | (Apomorphine) 6-Methyl-5,6,6a,...)
Affinity DataIC50: 384nMAssay Description:Compound was tested in vitro for binding affinity towards Dopamine receptor D1 in rat striatal membrane by using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007573(CHEMBL93428 | 4-(1-Propyl-1,2,5,6-tetrahydro-pyrid...)
Affinity DataIC50: 574nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 860nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 860nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007570(CHEMBL93972 | 7-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 1.13E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007575(CHEMBL328548 | 6-Propyl-4,5,5a,6,7,8,9,9a-octahydr...)
Affinity DataIC50: 1.24E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM81924(CAS_85976-54-1 | (R)-3-(1-Propyl-piperidin-3-yl)-p...)
Affinity DataIC50: 2.28E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007574(CHEMBL329444 | 7-Propyl-4,5,6,7,8,9-hexahydro-thia...)
Affinity DataIC50: 3.43E+3nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007575(CHEMBL328548 | 6-Propyl-4,5,5a,6,7,8,9,9a-octahydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM81924(CAS_85976-54-1 | (R)-3-(1-Propyl-piperidin-3-yl)-p...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007573(CHEMBL93428 | 4-(1-Propyl-1,2,5,6-tetrahydro-pyrid...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007574(CHEMBL329444 | 7-Propyl-4,5,6,7,8,9-hexahydro-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007570(CHEMBL93972 | 7-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007569(CHEMBL92784 | 8-Propyl-4,5,6,7,8,9-hexahydro-thiaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compound was tested in vitro for binding affinity against dopamine receptor D1 in rat striatal membrane by using DA antagonist [3H]NPAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity towards dopamine receptor D1 in rat striatal membrane using [3H]-SCH- 23390More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007571(CHEMBL91453 | 6-Propyl-4,5,5a,6,7,8-hexahydro-thia...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity towards dopamine receptor D1 in rat striatal membrane using [3H]-SCH- 23390More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007569(CHEMBL92784 | 8-Propyl-4,5,6,7,8,9-hexahydro-thiaz...)
Affinity DataIC50: 1.56E+4nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed