Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 50018033
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190203(2-amino-6-chloro-N-[8-chloro-11-(4-methyl-piperazi...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190049(2-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  1nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190193(naphthalene-1-carboxylic acid [8-chloro-11-(4-meth...)
Affinity DataKi:  1nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190186(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190059(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190062(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190186(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190203(2-amino-6-chloro-N-[8-chloro-11-(4-methyl-piperazi...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190208(2-amino-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-d...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190062(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190216(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190208(2-amino-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-d...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190187(2,6-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190202(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190193(naphthalene-1-carboxylic acid [8-chloro-11-(4-meth...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190049(2-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190214(3-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190205(2,4,6-trichloro-N-[8-chloro-11-(4-methyl-piperazin...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190186(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  7nMAssay Description:Binding affinity at dopamine D5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190192(2-amino-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-d...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190204(naphthalene-2-carboxylic acid [8-chloro-11-(4-meth...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190230(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190201(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190232(thiophene-3-carboxylic acid [8-chloro-11-(4-methyl...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190219(quinoline-2-carboxylic acid [8-chloro-11-(4-methyl...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190234(4-ethoxy-thiophene-2-carboxylic acid [8-chloro-11-...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190231(2-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190229(3,4-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190206(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190199(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190059(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  13.8nMAssay Description:Binding affinity at 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190207(4-bromo-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-d...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190226(thiophene-2-carboxylic acid [8-chloro-11-(4-methyl...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190189(furan-2-carboxylic acid [8-chloro-11-(4-methyl-pip...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190235(isoxazole-3-carboxylic acid [8-chloro-11-(4-methyl...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190209(isoquinoline-1-carboxylic acid [8-chloro-11-(4-met...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190195(3,5-dichloro-N-[8-chloro-11-(4-methyl-piperazin-1-...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190190(2-propyl-pentanoic acid [8-chloro-11-(4-methyl-pip...)
Affinity DataKi:  25.6nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190227(quinoline-3-carboxylic acid [8-chloro-11-(4-methyl...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190211(3-ethoxy-benzo[b]thiophene-2-carboxylic acid [8-ch...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190200(1-phenyl-5-trifluoromethyl-1H-pyrazole-4-carboxyli...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190062(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  31nMAssay Description:Binding affinity at dopamine D5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190221(4-chloro-N-[8-chloro-11-(4-methyl-piperazin-1-yl)-...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190059(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  38nMAssay Description:Binding affinity at dopamine D5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190191(3-phenyl-thiophene-2-carboxylic acid [8-chloro-11-...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190213(cyclohexanecarboxylic acid [8-chloro-11-(4-methyl-...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190215(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190057(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190233(N-[8-chloro-11-(4-methyl-piperazin-1-yl)-dibenzo[b...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1B) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50190203(2-amino-6-chloro-N-[8-chloro-11-(4-methyl-piperazi...)
Affinity DataKi:  53nMAssay Description:Binding affinity at dopamine D5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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