Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50037738
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 226nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat DAT expressed in D8 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(bip-tyr-thr-pro-thr(obzl)-gly | CHEMBL374492)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(bip-tyr-thr-pro-thr(obzl)-gly | CHEMBL374492)
Affinity DataIC50: 494nMAssay Description:Inhibition of [3H]WIN-35428 binding to rat DAT expressed in D8 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(bip-tyr-thr-ala-pro-phe | CHEMBL439332)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50084717(CHEMBL120901 | 3-Naphthalen-2-yl-8-oxa-bicyclo[3.2...)
Affinity DataIC50: 900nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190385(bip-tyr-thr-pro-ala-thr(obzl)-gly | CHEMBL219358)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190387(bip-tyr-thr-pro-lys-thr(obzl)-gly | CHEMBL428483)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190388(bip-tyr(3bzl)-thr-pro-lys-thr | CHEMBL385983)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190389(bip-tyr-ala-pro-lys-thr(obzl)-gly | CHEMBL277108)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(bip-tyr-thr-pro-lys-thr | CHEMBL379496)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190375(bip-tyr-thr(obzl)-pro-lys-thr-gly | CHEMBL269579)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(bip-tyr-thr-ala-pro-phe | CHEMBL439332)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(bip-tyr-thr-ala-pro-phe | CHEMBL439332)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(bip-tyr-thr-pro-thr(obzl)-gly | CHEMBL374492)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(bip-tyr-thr-pro-thr(obzl)-gly | CHEMBL374492)
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190376(bip-ala-thr-pro-lys-thr(obzl)-gly | CHEMBL383931)
Affinity DataIC50: 1.73E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190383(nal2-tyr-thr-pro-lys-thr(obzl)-gly | CHEMBL411570)
Affinity DataIC50: 1.84E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190384(nal1-tyr-thr-pro-lys-thr(obzl)-gly | CHEMBL218952)
Affinity DataIC50: 1.99E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190386(bpa-tyr-thr-pro-lys-thr(obzl)-gly | CHEMBL409615)
Affinity DataIC50: 2.39E+5nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(bip-tyr-thr-pro-lys-thr | CHEMBL379496)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190380(bip-tyr-thr-pro-thr(obzl)-gly | CHEMBL374492)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(bip-tyr-thr-pro-lys-thr | CHEMBL379496)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Mouse)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190379(bip-tyr-thr-ala-pro-phe | CHEMBL439332)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of mouse GAT1-mediated gamma-aminobutyric acid uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190381(bip-tyr-thr-ala-thr(obzl)-gly | CHEMBL209752)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190378(bip-tyr-thr-ala-lys-thr(obzl)-gly | CHEMBL219062)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190377(phe-phe-tyr-thr-pro-lys-thr | CHEMBL212513)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat DAT-mediated [3H]dopamine uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50190382(bip-tyr-thr-pro-lys-thr | CHEMBL379496)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of rat SERT-mediated serotonin uptake in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed