Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 4409
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68208(Type II inhibitor, 2)
Affinity DataIC50: 5nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68217(Type I progenitor, 11)
Affinity DataIC50: 5.70nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68217(Type I progenitor, 11)
Affinity DataIC50: 5.80nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM50242740(Type II inhibitor, 14 | CHEMBL459850 | N-(3-(7-Ami...)
Affinity DataIC50: 8nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68219(Type II inhibitor, 13)
Affinity DataIC50: 9.10nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM50242740(Type II inhibitor, 14 | CHEMBL459850 | N-(3-(7-Ami...)
Affinity DataIC50: 11nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68218(Type II inhibitor, 12)
Affinity DataIC50: 19.6nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM6568(PD-173955 | CHEMBL386051 | 6-(2,6-dichlorophenyl)-...)
Affinity DataIC50: 23nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM6568(PD-173955 | CHEMBL386051 | 6-(2,6-dichlorophenyl)-...)
Affinity DataIC50: 24nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 27nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68218(Type II inhibitor, 12)
Affinity DataIC50: 27.2nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68219(Type II inhibitor, 13)
Affinity DataIC50: 150nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68208(Type II inhibitor, 2)
Affinity DataIC50: 152nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68214(Type II inhibitor, 8)
Affinity DataIC50: 154nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68211(Type II inhibitor, 5)
Affinity DataIC50: 374nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68209(Type II inhibitor, 3)
Affinity DataIC50: 1.36E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68213(Type I progenitor, 7)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68207(Type I progenitor, 1)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68209(Type II inhibitor, 3)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68220(Type II inhibitor, 15)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68210(Type I progenitor, 4)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68211(Type II inhibitor, 5)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68212(Type II inhibitor, 6)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68213(Type I progenitor, 7)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68216(Type II inhibitor, 10)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68220(Type II inhibitor, 15)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68212(Type II inhibitor, 6)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68210(Type I progenitor, 4)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68214(Type II inhibitor, 8)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68207(Type I progenitor, 1)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using dephophorylated conformationally inactive Abl kinase was obtained by treating pure recombinant Abl with Yersinia ester...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM68216(Type II inhibitor, 10)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1 [1-999,Q252H](Human)
The Scripps Research Institute

LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataIC50: 5.00E+3nMpH: 7.5Assay Description:An in vitro kinase assay using phosphorylated recombinant human Abl kinase domains to phosphorylate a peptide substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/14/2011
Entry Details Article
PubMed