Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50018271
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193734(2-{[3-(4-methoxy-phenyl)-1-(3-trifluoromethyl-benz...)
Affinity DataIC50: 1nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193736(1-(3-(trifluoromethyl)benzyl)-3-(4-methoxyphenyl)-...)
Affinity DataIC50: 2nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193748(1-(3-(trifluoromethyl)benzyl)-3-(4-methoxyphenyl)-...)
Affinity DataIC50: 3nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193744(1-(3-(trifluoromethyl)benzyl)-N-(4-fluorophenylsul...)
Affinity DataIC50: 7nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193751(1-(3-(trifluoromethyl)benzyl)-3-(4-methoxyphenyl)-...)
Affinity DataIC50: 7nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193733(1-(3-(benzyloxy)benzyl)-N-(3-(trifluoromethyl)phen...)
Affinity DataIC50: 50nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193729(1-(3-(trifluoromethyl)benzyl)-3-(4-methoxyphenyl)-...)
Affinity DataIC50: 60nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193750(1-(3-(trifluoromethyl)benzyl)-N-(3-(trifluoromethy...)
Affinity DataIC50: 80nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193739(1-(3-(trifluoromethyl)benzyl)-N-(5-chlorothiophen-...)
Affinity DataIC50: 80nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193742(1-(3-(trifluoromethyl)benzyl)-N-(2-(trifluoromethy...)
Affinity DataIC50: 80nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193752(1-(3-(trifluoromethyl)benzyl)-N-(naphthalen-2-ylsu...)
Affinity DataIC50: 90nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataIC50: 90nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193741(1-(3-(trifluoromethoxy)benzyl)-N-(3-(trifluorometh...)
Affinity DataIC50: 90nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193735(1-(3-methoxybenzyl)-N-(3-(trifluoromethyl)phenylsu...)
Affinity DataIC50: 140nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193743(1-(3-(trifluoromethyl)benzyl)-N-(o-tolylsulfonyl)-...)
Affinity DataIC50: 180nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193745(1-(3-(trifluoromethyl)benzyl)-N-(4-chlorophenylsul...)
Affinity DataIC50: 280nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193754(1-benzyl-N-(3-(trifluoromethyl)phenylsulfonyl)-1H-...)
Affinity DataIC50: 280nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193728(1-(3-(trifluoromethyl)benzyl)-N-(phenylsulfonyl)-1...)
Affinity DataIC50: 290nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193727(1-(3-(trifluoromethyl)benzyl)-N-tosyl-1H-indole-2-...)
Affinity DataIC50: 290nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193747(1-(3-(trifluoromethyl)benzyl)-5-chloro-N-(3-(trifl...)
Affinity DataIC50: 330nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193732(1-(4-tert-butylbenzyl)-N-(3-(trifluoromethyl)pheny...)
Affinity DataIC50: 330nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193746(1-(2,5-dichlorobenzyl)-N-(3-(trifluoromethyl)pheny...)
Affinity DataIC50: 380nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193731(1-(4-(trifluoromethyl)benzyl)-N-(3-(trifluoromethy...)
Affinity DataIC50: 400nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193753(1-(3-(trifluoromethyl)benzyl)-5-hydroxy-N-(3-(trif...)
Affinity DataIC50: 540nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193740(1-(3-(trifluoromethyl)benzyl)-N-(methylsulfonyl)-1...)
Affinity DataIC50: 680nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193730(1-(4-(trifluoromethyl)benzyl)-N-(4-(trifluoromethy...)
Affinity DataIC50: 700nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193737(1-(3-(trifluoromethyl)benzyl)-N-(4-fluorophenylsul...)
Affinity DataIC50: 720nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193738(1-(3-(trifluoromethyl)benzyl)-5-(benzyloxy)-N-(3-(...)
Affinity DataIC50: 770nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193749(1-ethyl-N-(3-(trifluoromethyl)phenylsulfonyl)-1H-i...)
Affinity DataIC50: 2.44E+3nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Procter and Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50193755(1-(3-(trifluoromethyl)benzoyl)-N-(3-(trifluorometh...)
Affinity DataIC50: 9.40E+3nMAssay Description:Displacement of Fluormone from PPAR gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed