Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50018282
TargetTyrosine-protein kinase Yes(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 1nMAssay Description:Inhibition of YesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193891(US8481536, 577 | US8481536, 369 | CHEMBL218549 | 7...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193884(N-(4-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193879(US8481536, 364 | CHEMBL218656 | N-(4-(2-(diethylam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193910(US8481536, 370 | CHEMBL218102 | N-(3-(2-(diethylam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 13nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 20nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 21nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193897(7-(2,6-dimethylphenyl)-N-(4-(2-ethoxy-4-methylpipe...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Fyn(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 23nMAssay Description:Inhibition of FynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193881(N-(3-(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193903(7-(2,6-dimethylphenyl)-N-(4-(2-ethoxymorpholino)ph...)
Affinity DataIC50: 32nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193909(7-(2,6-dimethylphenyl)-5-methyl-N-(4-(4-methyl-2-p...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193890(7-(2,6-dimethylphenyl)-5-methyl-N-(3-(4-methyl-2-p...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193907(US8481536, 359 | CHEMBL221582 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193877(7-(2,6-dimethylphenyl)-N-(3-(2-ethoxy-4-methylpipe...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEphrin type-B receptor 4(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 64nMAssay Description:Inhibition of EphB4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 68nMAssay Description:Inhibition of Raf1 kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193902(US8481536, 345 | CHEMBL221431 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193908(CHEMBL218281 | US8481536, 426 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 128nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193887(CHEMBL221975 | US8481536, 320 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193892(US8481536, 346 | CHEMBL217961 | N-(3-chlorophenyl)...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193915(CHEMBL446951 | US8481536, 415 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 137nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193885(CHEMBL220798 | US8481536, 344 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193886(US8481536, 585 | US8481536, 397 | CHEMBL218597 | 3...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193898(US8481536, 332 | CHEMBL218742 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 180nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193882(CHEMBL220912 | US8481536, 375 | N1-(7-(2,6-dimethy...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193894(CHEMBL436516 | US8481536, 408 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193889(US8481536, 573 | CHEMBL374248 | US8481536, 316 | 7...)
Affinity DataIC50: 410nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193901(US8481536, 422 | CHEMBL218049 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 555nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase CSK(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 659nMAssay Description:Inhibition of CSKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiopoietin-1 receptor(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 678nMAssay Description:Inhibition of Tie2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 960nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193873(US8481536, 337 | CHEMBL220480 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 960nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 965nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of BlkMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193904(3-(3-amino-5-methylbenzo[e][1,2,4]triazin-7-yl)-4-...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193883(CHEMBL218042 | US8481536, 572 | US8481536, 314 | 7...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193880(CHEMBL218598 | US8481536, 328 | N-(7-(2,6-dimethyl...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193899(7-(2,6-dimethylphenyl)benzo[e][1,2,4]triazin-3-ami...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase beta-1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of p70S6KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193916(7-(2,6-dichlorophenyl)-5-methylbenzo[e][1,2,4]tria...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193895(7-(naphthalen-2-yl)benzo[e][1,2,4]triazin-3-amine ...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193874(CHEMBL436137 | US8481536, 322 | 7-(2,6-dimethylphe...)
Affinity DataIC50: 5.99E+3nMAssay Description:Inhibition of Abl T315I mutantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193913(7-(2,6-dimethylphenyl)-5-methylbenzo[e][1,2,4]tria...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193912(7-(benzo[d][1,3]dioxol-5-yl)benzo[e][1,2,4]triazin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Targegen

Curated by ChEMBL
LigandPNGBDBM50193876(3-(3-aminobenzo[e][1,2,4]triazin-7-yl)phenol | CHE...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human recombinant Src kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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