Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50018332
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194487(3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropy...)
Affinity DataIC50: 1.79nMAssay Description:Activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194488(6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropy...)
Affinity DataIC50: 4.93nMAssay Description:Activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194487(3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropy...)
Affinity DataIC50: 25.8nMAssay Description:Activity at delta opioid receptor assessed as inhibition of muscle contraction in mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194488(6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Activity at delta opioid receptor assessed as inhibition of muscle contraction in mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194487(3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropy...)
Affinity DataKi:  0.0210nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194488(6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropy...)
Affinity DataKi:  0.0510nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194490(3-[4'-(H-Tyr)-aminobutyl]-6-[3'-(H-Tyr)-amino-prop...)
Affinity DataKi:  7.58nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194488(6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropy...)
Affinity DataKi:  18.8nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194489(6-[4'-(H-Tyr)-aminobutyl]-3-[3'-(H-tyr)-amino-prop...)
Affinity DataKi:  27.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194487(3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropy...)
Affinity DataKi:  31.9nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194490(3-[4'-(H-Tyr)-aminobutyl]-6-[3'-(H-Tyr)-amino-prop...)
Affinity DataKi:  924nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50194489(6-[4'-(H-Tyr)-aminobutyl]-3-[3'-(H-tyr)-amino-prop...)
Affinity DataKi:  2.77E+3nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed