Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50018554
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197001(N-[2'-(isoxazol-5-ylsulfamoyl)-4-oxazol-2-yl-biphe...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197003(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-(2-{2-[2-({[2'-(i...)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197002(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-{2-[2-(2-{2-[4-({...)
Affinity DataIC50: 4.60nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197000(N-(35-{[4-(3,5-dioxohexyl)phenyl]carbamoyl}-3,6,9,...)
Affinity DataIC50: 7.70nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197004(3-{2-[2-(2-{2-[2-(2-{2-[4-(3,5-dioxo-hexyl)-phenyl...)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50196999(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-{2-[2-(2-{2-[4-(2...)
Affinity DataIC50: 21.6nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197005(N-[4-{2-[2-(2-{2-[4-(3,5-dioxo-hexyl)-phenylcarbam...)
Affinity DataIC50: 44.9nMAssay Description:Displacement of [125I]ET1 from human ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197003(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-(2-{2-[2-({[2'-(i...)
Affinity DataIC50: 1.11E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197002(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-{2-[2-(2-{2-[4-({...)
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197000(N-(35-{[4-(3,5-dioxohexyl)phenyl]carbamoyl}-3,6,9,...)
Affinity DataIC50: 4.51E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197004(3-{2-[2-(2-{2-[2-(2-{2-[4-(3,5-dioxo-hexyl)-phenyl...)
Affinity DataIC50: 4.69E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50196999(N-[4-(3,5-dioxo-hexyl)-phenyl]-3-{2-[2-(2-{2-[4-(2...)
Affinity DataIC50: 4.92E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197001(N-[2'-(isoxazol-5-ylsulfamoyl)-4-oxazol-2-yl-biphe...)
Affinity DataIC50: 6.00E+3nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Covx Research

Curated by ChEMBL
LigandPNGBDBM50197005(N-[4-{2-[2-(2-{2-[4-(3,5-dioxo-hexyl)-phenylcarbam...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed