Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50025072
TargetNeuronal acetylcholine receptor subunit alpha-3(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241747(3-demethoxy-2alpha,3alpha-methylenedioxyerythrocul...)
Affinity DataIC50: 7.70E+4nMAssay Description:Antagonist activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha-3-beta-4R2 cells assessed as nicotine-induced calcium fluorescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241746(15-amido-3-demethoxy-2alpha,3alpha-methylenedioxye...)
Affinity DataIC50: 9.40E+4nMAssay Description:Antagonist activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha-3-beta-4R2 cells assessed as nicotine-induced calcium fluorescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Rat)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50241748(dihydro-beta-erythroidine | CHEMBL518059)
Affinity DataIC50: 1.00E+5nMAssay Description:Activity at rat alpha3beta4 nicotinic receptor expressed in KXalpha-3-beta-4R2 cells assessed as nicotine-induced 86Rb+ effluxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed