Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50042260
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423023(CHEMBL427844)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423034(CHEMBL390189)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423041(CHEMBL430360)
Affinity DataIC50: 0.790nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423044(CHEMBL234519)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423042(CHEMBL390238)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423032(CHEMBL234727)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423033(CHEMBL428367)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423019(CHEMBL390038)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423026(CHEMBL234945)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423043(CHEMBL234946)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423037(CHEMBL234518)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423023(CHEMBL427844)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of TP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423018(CHEMBL390190)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423039(CHEMBL234302)
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423038(CHEMBL234301)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423015(CHEMBL234721)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423031(CHEMBL234303)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423027(CHEMBL389995)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423020(CHEMBL388242)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423028(CHEMBL390660)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423021(CHEMBL234722)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423022(CHEMBL234728)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423017(CHEMBL395523)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50187023(3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methy...)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423035(CHEMBL395310)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423036(CHEMBL266258)
Affinity DataIC50: 6.30nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423025(CHEMBL388038)
Affinity DataIC50: 7.90nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423029(CHEMBL429259)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423016(CHEMBL388243)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423040(CHEMBL233872)
Affinity DataIC50: 126nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP4 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423023(CHEMBL427844)
Affinity DataIC50: 158nMAssay Description:Inhibition of EP4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423030(CHEMBL395756)
Affinity DataIC50: 158nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423014(CHEMBL233871)
Affinity DataIC50: 251nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP1 subtype(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423024(CHEMBL233665)
Affinity DataIC50: 316nMAssay Description:Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed