Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50018870
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 0.270nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 4.03nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 6.88nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataIC50: 283nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataIC50: 344nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199867((S)-2-allylamino-N-(5-{[(S)-2-allylamino-3-(4-hydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199867((S)-2-allylamino-N-(5-{[(S)-2-allylamino-3-(4-hydr...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199859((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199863((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199864((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199863((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199859((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199862((S)-2-allylamino-N-{6-[(S)-2-allylamino-3-(4-hydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199861((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199864((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199861((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199862((S)-2-allylamino-N-{6-[(S)-2-allylamino-3-(4-hydro...)
Affinity DataIC50: 1.00E+4nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataKi:  0.0540nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199863((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199861((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataKi:  1.33nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199859((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199867((S)-2-allylamino-N-(5-{[(S)-2-allylamino-3-(4-hydr...)
Affinity DataKi:  6.94nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199863((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  10.3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199862((S)-2-allylamino-N-{6-[(S)-2-allylamino-3-(4-hydro...)
Affinity DataKi:  12.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199864((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  13.1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199862((S)-2-allylamino-N-{6-[(S)-2-allylamino-3-(4-hydro...)
Affinity DataKi:  51.5nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199867((S)-2-allylamino-N-(5-{[(S)-2-allylamino-3-(4-hydr...)
Affinity DataKi:  77.8nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199860((S)-1-((S)-2-(allylamino)-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199859((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  217nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199861((S)-1-((S)-2-(allylamino)-3-(4-hydroxy-2,6-dimethy...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199866((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199864((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  1.42E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50095155(CHEMBL316446 | (S)-1-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199866((S)-N-((S)-1-((S)-1-(allylamino)-1-oxo-3-phenylpro...)
Affinity DataKi:  5.76E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50139013(CHEMBL333357 | (S)-N-((S)-1-((S)-1-amino-1-oxo-3-p...)
Affinity DataKi:  6.08E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199860((S)-1-((S)-2-(allylamino)-3-(4-hydroxyphenyl)propa...)
Affinity DataKi:  7.36E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed