Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 2620
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22714(N-[(4-fluorophenyl)methyl]-5,6-dihydroxy-2-(thioph...)
Affinity DataIC50: 10nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22717(2-benzyl-N-[(4-fluorophenyl)methyl]-5,6-dihydroxyp...)
Affinity DataIC50: 50nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22720(2-[2-(dimethylamino)propan-2-yl]-N-[(4-fluoropheny...)
Affinity DataIC50: 50nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22663(N-[(4-fluorophenyl)methyl]-5,6-dihydroxypyrimidine...)
Affinity DataIC50: 60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22715(N-[(4-fluorophenyl)methyl]-5,6-dihydroxy-2-methylp...)
Affinity DataIC50: 60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22628(N-[(4-fluorophenyl)methyl]-5-hydroxy-1-methyl-2-(3...)
Affinity DataIC50: 60nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22716(N-benzyl-5,6-dihydroxy-2-phenylpyrimidine-4-carbox...)
Affinity DataIC50: 70nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22664(JMC496646 Compound 11 | 2-[1-(dimethylamino)ethyl]...)
Affinity DataIC50: 80nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22713(N-benzyl-5,6-dihydroxy-2-(thiophen-2-yl)pyrimidine...)
Affinity DataIC50: 85nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22718(2-[(dimethylamino)(phenyl)methyl]-N-[(4-fluorophen...)
Affinity DataIC50: 200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22719(2-[(dimethylamino)methyl]-N-[(4-fluorophenyl)methy...)
Affinity DataIC50: 200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22609(JMC496646 Compound 14 | N-[(4-fluorophenyl)methyl]...)
Affinity DataIC50: 200nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Irbm-Mrl

LigandPNGBDBM22611(JMC496646 Compound 16 | N-[(4-fluorophenyl)methyl]...)
Affinity DataIC50: 210nMpH: 7.8 T: 2°CAssay Description:The microtiter plate assay for stand transfer was performed with an immobilized donor substrate and a target substrate biotinylated at the 3-prime en...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2008
Entry Details Article
PubMed