Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50019060
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201230(4-(2,4-dichloro-5-methoxyphenylamino)-6-ethoxy-7-(...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201234(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201232(4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-(dimeth...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201226(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201236(4-(2,4-dichlorophenylamino)-6-methoxy-7-(4-(4-meth...)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201229(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201228(6-methoxy-7-(4-(4-methylpiperazin-1-yl)but-1-ynyl)...)
Affinity DataIC50: 21nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201233(4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-(4-meth...)
Affinity DataIC50: 28nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 73nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201230(4-(2,4-dichloro-5-methoxyphenylamino)-6-ethoxy-7-(...)
Affinity DataIC50: 130nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201234(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201235(7-(4-(4-methylpiperazin-1-yl)but-1-ynyl)-4-(3,4,5-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201231(4-(2,4-dichloro-5-methoxyphenylamino)-6-(4-(4-meth...)
Affinity DataIC50: 230nMAssay Description:Inhibition of Src activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201232(4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-(dimeth...)
Affinity DataIC50: 250nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201236(4-(2,4-dichlorophenylamino)-6-methoxy-7-(4-(4-meth...)
Affinity DataIC50: 430nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201226(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 520nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201228(6-methoxy-7-(4-(4-methylpiperazin-1-yl)but-1-ynyl)...)
Affinity DataIC50: 590nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 720nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201229(4-(2,4-dichloro-5-methoxyphenylamino)-6-methoxy-7-...)
Affinity DataIC50: 740nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201233(4-(2,4-dichloro-5-methoxyphenylamino)-7-(4-(4-meth...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201235(7-(4-(4-methylpiperazin-1-yl)but-1-ynyl)-4-(3,4,5-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201231(4-(2,4-dichloro-5-methoxyphenylamino)-6-(4-(4-meth...)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of Src in rat fibroblastsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of AKTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50201227(4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of CDK4More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed