Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 2563
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22038(2-[2-(4-fluorophenyl)-1H-indol-3-yl]-N,N-dihexyl-2...)
Affinity DataKi:  0.370nM ΔG°:  -50.0kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22041(2-[6-chloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridi...)
Affinity DataKi:  0.5nM ΔG°:  -49.3kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22032(PK 11195 | PK11195 | RP 52028 | N-(butan-2-yl)-1-(...)
Affinity DataKi:  9.30nM ΔG°:  -42.6kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22037(2-[2-(4-fluorophenyl)-1H-indol-3-yl]-N-{6-[(7-nitr...)
Affinity DataKi:  12nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22036(7-nitrobenz-2-oxa-1,3-diazol-4-yl (NBD)-group cont...)
Affinity DataKi:  17nM ΔG°:  -41.2kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22035(2-[2-(4-fluorophenyl)-1H-indol-3-yl]-N-{4-[(7-nitr...)
Affinity DataKi:  23nM ΔG°:  -40.5kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22040(Ro5-4864 | 4' Cl-diazepam | 4 -chlorodiazepam ...)
Affinity DataKi:  23nM ΔG°:  -40.5kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22034(N-{4-[(7-nitro-2,1,3-benzoxadiazol-4-yl)amino]buty...)
Affinity DataKi:  42nM ΔG°:  -39.1kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22033(2-[2-(4-fluorophenyl)-1H-indol-3-yl]-N-{2-[(7-nitr...)
Affinity DataKi:  835nM ΔG°:  -32.2kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita Di Pisa

LigandPNGBDBM22031(N-{2-[(7-nitro-2,1,3-benzoxadiazol-4-yl)amino]ethy...)
Affinity DataKi:  994nM ΔG°:  -31.8kJ/molepH: 7.4 T: 2°CAssay Description:Assays were performed by incubating aliquots of rat kidney mitochondria suspensions with [3H]PK 11195 and a range of concentrations of the test compo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2008
Entry Details Article
PubMed