Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50019273
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203383(N-(1-benzylpiperidine-4-yl)-2-naphthamide | N-(1-b...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203374(naphthalene-2-carboxylic acid [1-(3-methyl-benzyl)...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203397(N-(1-(3-methoxybenzyl)piperidin-4-yl)-2-naphthamid...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203376(naphthalene-2-carboxylic acid [1-(4-methyl-benzyl)...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203377(naphthalene-2-carboxylic acid [1-(2-methyl-benzyl)...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203392(N-(1-(4-methoxybenzyl)piperidin-4-yl)-2-naphthamid...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203373(N-(1-(4-bromobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203382(N-(1-(3-bromobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203378(N-(1-(4-chlorobenzyl)piperidin-4-yl)-2-naphthamide...)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203388(N-(1-(4-chlorobenzyl)piperidin-4-yl)-1-naphthamide...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203394(N-(1-(4-bromobenzyl)piperidin-4-yl)-1-naphthamide ...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203383(N-(1-benzylpiperidine-4-yl)-2-naphthamide | N-(1-b...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203382(N-(1-(3-bromobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203389(N-(1-(3-chlorobenzyl)piperidin-4-yl)-2-naphthamide...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203393(N-(1-(3-bromobenzyl)piperidin-4-yl)-1-naphthamide ...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203391(naphthalene-1-carboxylic acid [1-(4-methyl-benzyl)...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203384(naphthalene-1-carboxylic acid [1-(3-methyl-benzyl)...)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203386(N-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yl)-2-...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203374(naphthalene-2-carboxylic acid [1-(3-methyl-benzyl)...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203385(N-(1-(4-(trifluoromethyl)benzyl)piperidin-4-yl)-1-...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203381(N-(1-(3-(trifluoromethyl)benzyl)piperidin-4-yl)-2-...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203398(N-(1-(3-chlorobenzyl)piperidin-4-yl)-1-naphthamide...)
Affinity DataKi:  116nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203371(N-(1-(3-(trifluoromethyl)benzyl)piperidin-4-yl)-1-...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203399(N-(1-(2-chlorobenzyl)piperidin-4-yl)-2-naphthamide...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203389(N-(1-(3-chlorobenzyl)piperidin-4-yl)-2-naphthamide...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203392(N-(1-(4-methoxybenzyl)piperidin-4-yl)-2-naphthamid...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203372(naphthalene-1-carboxylic acid [1-(2-methyl-benzyl)...)
Affinity DataKi:  155nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203397(N-(1-(3-methoxybenzyl)piperidin-4-yl)-2-naphthamid...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203375(N-(1-benzylpiperidine-4-yl)-1-naphthamide | N-(1-b...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203379(N-(1-(3-methoxybenzyl)piperidin-4-yl)-1-naphthamid...)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203377(naphthalene-2-carboxylic acid [1-(2-methyl-benzyl)...)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203395(N-(1-(4-nitrobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203376(naphthalene-2-carboxylic acid [1-(4-methyl-benzyl)...)
Affinity DataKi:  222nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203396(N-(1-(4-methoxybenzyl)piperidin-4-yl)-1-naphthamid...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203373(N-(1-(4-bromobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  223nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203380(N-(1-(perfluorobenzyl)piperidin-4-yl)-1-naphthamid...)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203378(N-(1-(4-chlorobenzyl)piperidin-4-yl)-2-naphthamide...)
Affinity DataKi:  242nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203395(N-(1-(4-nitrobenzyl)piperidin-4-yl)-2-naphthamide ...)
Affinity DataKi:  278nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203370(N-(1-(pyridin-2-ylmethyl)piperidin-4-yl)-2-naphtha...)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203390(N-(1-(pyridin-3-ylmethyl)piperidin-4-yl)-2-naphtha...)
Affinity DataKi:  326nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(4) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203400(N-(1-(2-chlorobenzyl)piperidin-4-yl)-1-naphthamide...)
Affinity DataKi:  329nMAssay Description:Displacement of [3H]nemonapride from human cloned dopamine D4.2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203393(N-(1-(3-bromobenzyl)piperidin-4-yl)-1-naphthamide ...)
Affinity DataKi:  462nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203390(N-(1-(pyridin-3-ylmethyl)piperidin-4-yl)-2-naphtha...)
Affinity DataKi:  524nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203370(N-(1-(pyridin-2-ylmethyl)piperidin-4-yl)-2-naphtha...)
Affinity DataKi:  545nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203387(N-(1-(pyridin-4-ylmethyl)piperidin-4-yl)-2-naphtha...)
Affinity DataKi:  695nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203383(N-(1-benzylpiperidine-4-yl)-2-naphthamide | N-(1-b...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Université

Curated by ChEMBL
LigandPNGBDBM50203375(N-(1-benzylpiperidine-4-yl)-1-naphthamide | N-(1-b...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from rat 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50203375(N-(1-benzylpiperidine-4-yl)-1-naphthamide | N-(1-b...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from human cloned dopamine D2L receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed