Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50037831
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204623([2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204626((2-(hydroxymethyl)-5-oxo-4-(propan-2-ylidene)-tetr...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204628([2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204630([2-(hydroxymethyl)-4-(methylethylidene)-5-oxo-2-2,...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204629(methyl 2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)-4-(me...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50370871(CHEMBL1162941)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204625(methyl 16-{4-[2-(4-{2-[4-({[2-(Hydroxymethyl)-4-(m...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204624(tert-butyl 2-({[(tert-Butyl)oxycarbonyl]methyl}{2-...)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204622(methyl 2-[4-(2-{4-[2-(4-{2-[4-({[2-(hydroxymethyl)...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50204627(2-(N-(carboxymethyl){2-[2-(2-{4-[2-(4-{2-[4-({[2-(...)
Affinity DataKi:  1.39E+3nMAssay Description:Displacement of [3H]PDBu from PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed