Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019518
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205442(2-thiosalvinorin B | CHEMBL231536)
Affinity DataEC50:  287nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  2.82nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205443(2-epi-2-thiosalvinorin A | CHEMBL231537)
Affinity DataEC50:  123nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205444(2-epi-2-thiosalvinorin B | CHEMBL231638)
Affinity DataEC50: >2.00E+3nMAssay Description:Activity at human kappa opioid receptor expressed in HEK293 cells as intracellular calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataKi:  0.75nMAssay Description:Displacement of [3H]U-69593 from rat cloned KORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205442(2-thiosalvinorin B | CHEMBL231536)
Affinity DataKi:  54.5nMAssay Description:Displacement of [3H]U-69593 from rat cloned KORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205443(2-epi-2-thiosalvinorin A | CHEMBL231537)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]U-69593 from rat cloned KORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Rat)
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50205444(2-epi-2-thiosalvinorin B | CHEMBL231638)
Affinity DataKi:  546nMAssay Description:Displacement of [3H]U-69593 from rat cloned KORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed