Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50019574
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 0.275nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 0.496nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 | CHEMBL220327)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 | CHEMBL220327)
Affinity DataIC50: 0.562nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205830(H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 | CHEMBL373572)
Affinity DataIC50: 0.603nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  0.616nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 | CHEMBL220327)
Affinity DataKi:  0.822nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 0.898nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 | CHEMBL...)
Affinity DataIC50: 1.02nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  1.05nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205833(H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  1.17nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  1.25nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 | CHEMBL220327)
Affinity DataIC50: 1.30nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205830(H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 | CHEMBL373572)
Affinity DataKi:  1.61nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205830(H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 | CHEMBL373572)
Affinity DataIC50: 1.65nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205830(H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 | CHEMBL373572)
Affinity DataKi:  1.74nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 1.81nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  1.92nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  2.27nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  2.34nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]DAMGO from rat brain mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 | CHEMBL...)
Affinity DataIC50: 3.19nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205833(H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  3.34nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205833(H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 | CHEMBL...)
Affinity DataIC50: 3.64nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 4.38nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 5.63nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  5.87nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  6.55nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  7.04nMAssay Description:Displacement of [3H]DSLET from rat brain delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 9.91nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205833(H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 | CHEMBL...)
Affinity DataIC50: 11.2nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataIC50: 11.9nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  30.4nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205830(H-Tyr-c[D-Cys-Gly-Phe-L-Cys]NH2 | CHEMBL373572)
Affinity DataKi:  40.1nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205832(H-Tyr-c[D-Cys-Gly-Phe-D-Cys]NH2 | CHEMBL220327)
Affinity DataKi:  44.9nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  57.6nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205833(H-Tyr-c[D-Allylgly-Gly-Phe-D-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  71.5nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205834(CHEMBL223244 | CHEMBL220333 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205831(H-Tyr-c[D-Allylgly-Gly-Phe-L-Allylgly]NH2 | CHEMBL...)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Clinical Research Institute of Montreal

Curated by ChEMBL
LigandPNGBDBM50205828(CHEMBL220219 | CHEMBL373796 | H-Tyr-c[D-Allylgly-G...)
Affinity DataKi:  498nMAssay Description:Displacement of [3H]U-69593 from guinea pig brain kappa opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed