Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50037936
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371107(CHEMBL397235)
Affinity DataIC50: 350nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50206310(ELACRIDAR HYDROCHLORIDE | N-4-[2-(1,2,3,4-Tetrahyd...)
Affinity DataIC50: 410nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371104(CHEMBL243167)
Affinity DataIC50: 450nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371110(CHEMBL243168)
Affinity DataIC50: 560nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371108(CHEMBL242513)
Affinity DataIC50: 770nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371114(CHEMBL243169)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371109(GNF-PF-2549 | CHEMBL388886)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371106(CHEMBL243813)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371105(CHEMBL243814)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371103(CHEMBL242942)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM60916(2-oxidanyl-10H-acridin-9-one | MLS001179906 | cid_...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371111(CHEMBL397685)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371112(CHEMBL242943)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Human)
Umr 5063 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50371113(CHEMBL242512)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of ABCG2 expressed in HEK293 cells assessed as mitoxantrone-mediated efflux by flow cytometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2012
Entry Details Article
PubMed