Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50048883
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230008(CHEMBL318528)
Affinity DataKd:  1.52E+4nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230009(CHEMBL97915)
Affinity DataKd:  100nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50227330(CHEMBL420268)
Affinity DataKd:  150nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKd:  0.900nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004734(CHEMBL310852 | N-Methyl-N-(1-methyl-4-pyrrolidin-1...)
Affinity DataKd:  240nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004726(CHEMBL51682 | 1-(1-Methyl-4-pyrrolidin-1-yl-but-2-...)
Affinity DataKd:  91nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230010(CHEMBL319665)
Affinity DataKd:  5.89E+3nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230006(CHEMBL99266)
Affinity DataKd:  500nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230000(CHEMBL99265)
Affinity DataKd:  2.05E+4nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230003(CHEMBL97890)
Affinity DataKd:  8.10E+3nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230011(CHEMBL100406)
Affinity DataKd:  620nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230002(CHEMBL318049)
Affinity DataKd:  850nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230004(CHEMBL101645)
Affinity DataKd:  200nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230007(CHEMBL101646)
Affinity DataKd:  1.12E+4nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Human)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50228614(CHEMBL51405)
Affinity DataKd:  93nMAssay Description:Determination of dissociation constant from antimuscarinic activity on isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50228614(CHEMBL51405)
Affinity DataKi:  56nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50004734(CHEMBL310852 | N-Methyl-N-(1-methyl-4-pyrrolidin-1...)
Affinity DataKi:  64nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230004(CHEMBL101645)
Affinity DataKi:  110nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230009(CHEMBL97915)
Affinity DataKi:  120nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230006(CHEMBL99266)
Affinity DataKi:  230nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230011(CHEMBL100406)
Affinity DataKi:  310nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230002(CHEMBL318049)
Affinity DataKi:  540nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230010(CHEMBL319665)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230003(CHEMBL97890)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230000(CHEMBL99265)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230008(CHEMBL318528)
Affinity DataKi:  5.77E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Uppsala

Curated by ChEMBL
LigandPNGBDBM50230007(CHEMBL101646)
Affinity DataKi:  6.91E+3nMAssay Description:Inhibition of [3H]N-methylscopolamine binding to muscarinic acetylcholine receptor of rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed