Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50037908
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kc2betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207163(4-morpholin-4-yl-2-[3-(2-morpholin-4-yl-ethoxy)-ph...)
Affinity DataIC50: 16nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207172([3-(4-morpholin-4-yl-pyrido[3',2':4,5]furo[3,2-d]p...)
Affinity DataIC50: 24nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207169(4-(4-morpholin-4-yl-pyrido[3',2':4,5]furo[3,2-d]py...)
Affinity DataIC50: 26nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207173(4-morpholin-4-yl-2-[3-(2-thiomorpholin-4-yl-ethoxy...)
Affinity DataIC50: 79nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207170(2-(3-methoxy-phenyl)-4-morpholin-4-yl-pyrido[3',2'...)
Affinity DataIC50: 100nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207167(3-(4-morpholin-4-yl-pyrido[3',2':4,5]furo[3,2-d]py...)
Affinity DataIC50: 140nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207165(4-morpholin-4-yl-2-phenyl-pyrido[3',2':4,5]furo[3,...)
Affinity DataIC50: 160nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207175(4-morpholin-4-yl-2-[3-(2-piperidin-1-yl-ethoxy)-ph...)
Affinity DataIC50: 170nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 220nMAssay Description:Inhibition of PI3Kc2betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 340nMAssay Description:Inhibition of p110betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207168(2-(4-morpholin-4-yl-pyrido[3',2':4,5]furo[3,2-d]py...)
Affinity DataIC50: 400nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207178(4-morpholin-4-yl-pyrido[3',2':4,5]furo[3,2-d]pyrim...)
Affinity DataIC50: 560nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 630nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 660nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207177(4-morpholin-4-yl-pyrido[3',2':4,5]thieno[3,2-d]pyr...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p110gammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207176(4-morpholin-4-yl-2-phenyl-pyrido[3',2':4,5]thieno[...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM12915(CHEMBL98350 | 2-(morpholin-4-yl)-8-phenyl-4H-chrom...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PI3Kc2betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207174(4-morpholin-4-yl-benzo[4,5]thieno[3,2-d]pyrimidine...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Cyclin E/CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207179(8-morpholin-4-yl-9H-1,5,7,9-tetraaza-fluorene | CH...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM50207171(4-morpholin-4-yl-2-phenyl-benzo[4,5]thieno[3,2-d]p...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of p110alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of KDRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Cyclin E/CDK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 4.66E+5nMAssay Description:Inhibition of PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed