Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 2160
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17617(6-[(4-fluorobenzene)sulfonamido]-3-(furan-3-yl)-2-...)
Affinity DataIC50: 8nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17630(6-[(2-{[4-(dimethylamino)butyl]amino}benzene)sulfo...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17616(3-ethyl-6-[(4-fluorobenzene)sulfonamido]-2-methoxy...)
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17622(2-chloro-3-ethyl-6-[(4-fluorobenzene)sulfonamido]b...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17635(6-({2-[(1Z)-3-(diethylamino)prop-1-en-1-yl]-4-fluo...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17632(3-ethyl-2-methoxy-6-[(2-{[2-(1-methylpyrrolidin-2-...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17611(3-ethyl-6-[(4-fluorobenzene)sulfonamido]-2-methylb...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17627(2-(2-aminoethoxy)-3-ethyl-6-[(2-propylbenzene)sulf...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17634(6-[(2-{[3-(dimethylamino)propyl]amino}-4-fluoroben...)
Affinity DataIC50: 17nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17631(3-ethyl-2-methoxy-6-[(2-{[3-(2-methylpiperidin-1-y...)
Affinity DataIC50: 18nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17618(6-[(2-bromo-4-fluorobenzene)sulfonamido]-3-(furan-...)
Affinity DataIC50: 20nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17629(2-(2-aminoethoxy)-6-({2-[3-(diethylamino)propyl]-4...)
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17633(6-({2-[(1Z)-3-(diethylamino)prop-1-en-1-yl]-4-fluo...)
Affinity DataIC50: 26nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17624(2-ethoxy-3-ethyl-6-[(4-fluorobenzene)sulfonamido]b...)
Affinity DataIC50: 38nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17625(2-(2-aminoethoxy)-3-ethyl-6-[(4-fluorobenzene)sulf...)
Affinity DataIC50: 46nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17623(5-ethyl-2-[(4-fluorobenzene)sulfonamido]benzoic ac...)
Affinity DataIC50: 55nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17610(3-ethenyl-6-[(4-fluorobenzene)sulfonamido]-2-methy...)
Affinity DataIC50: 60nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17628(3-ethyl-2-methyl-6-(pyridine-2-sulfonamido)benzoic...)
Affinity DataIC50: 67nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17609(6-[(4-fluorobenzene)sulfonamido]-2,3-dimethylbenzo...)
Affinity DataIC50: 78nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17612(6-[(4-fluorobenzene)sulfonamido]-2-methyl-3-propyl...)
Affinity DataIC50: 150nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17621(6-[(4-fluorobenzene)sulfonamido]-2-methoxy-3-(1H-p...)
Affinity DataIC50: 280nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17619(6-[(2-bromo-4-fluorobenzene)sulfonamido]-3-(furan-...)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17613(3-butyl-6-[(4-fluorobenzene)sulfonamido]-2-methylb...)
Affinity DataIC50: 1.30E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17615(6-[(4-fluorobenzene)sulfonamido]-3-(1-hydroxyethyl...)
Affinity DataIC50: 2.50E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17626(2-(carboxymethoxy)-3-ethyl-6-[(4-fluorobenzene)sul...)
Affinity DataIC50: 5.80E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17614(6-[(4-fluorobenzene)sulfonamido]-3-(hydroxymethyl)...)
Affinity DataIC50: 8.00E+3nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed
TargetMethionine aminopeptidase 2(Human)
Abbott Laboratories

LigandPNGBDBM17620(6-[(2-bromo-4-fluorobenzene)sulfonamido]-3-(1H-imi...)
Affinity DataIC50: 3.60E+4nMpH: 7.4 T: 2°CAssay Description:A coupled enzyme chromogenic assay was developed to measure methionine aminopeptidase-2 activity by monitoring the production of free methionine with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2007
Entry Details Article
PubMed