Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50037875
TargetDelta-type opioid receptor(Mouse)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  14.9nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  26.2nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM21864(NALTRINDOLE | (8R)-7-(cyclopropylmethyl)-5,6,7,8,1...)
Affinity DataKi:  33.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209644(17-cyclopropylmethyl)-6,7-didehydro-4,5alpha-epoxy...)
Affinity DataKi:  48.2nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  1.75E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Missouri-Columbia

Curated by ChEMBL
LigandPNGBDBM50209645(17-(cyclopropylmethyl)-6,7-didehydro-4,5alpha-epox...)
Affinity DataKi:  2.01E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2012
Entry Details Article
PubMed