Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50020065
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50196898(((2R,6S)-1-(4-chlorophenylsulfonyl)-6-phenylpiperi...)
Affinity DataIC50: 16nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210042(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 60nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50196629((1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroquin...)
Affinity DataIC50: 73nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210040(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 86nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210044(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 120nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210041(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 140nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210043(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 180nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210045(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 180nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210027(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 190nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210033(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 220nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210028(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 280nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210039(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 360nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210046(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 450nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210036(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 530nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210032(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 540nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210034(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 600nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210026(((2R,5S)-1-(4-chlorophenylsulfonyl)-5-phenylpyrrol...)
Affinity DataIC50: 650nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210030(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 680nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210038(3-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 780nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210037(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 880nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210029(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 900nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210035(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Pharmacopeia Drug Discovery

Curated by ChEMBL
LigandPNGBDBM50210031(2-(1-(4-chlorophenylsulfonyl)-1,2,3,4-tetrahydroqu...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of gamma-secretaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed