Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 2996
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26758(2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imid...)
Affinity DataIC50: 2nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26759(2-fluorophenyl N-[7-(2-methyl-4,5-diphenyl-1H-imid...)
Affinity DataIC50: 4.20nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26757(phenyl N-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1-y...)
Affinity DataIC50: 5.30nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26766(2-fluorophenyl N-{6-[4,5-bis(4-fluorophenyl)-2-met...)
Affinity DataIC50: 10nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26748(CHEMBL237044 | ethyl 7-(2-ethyl-4,5-diphenyl-1H-im...)
Affinity DataIC50: 11nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26767(2,6-difluorophenyl N-{6-[4,5-bis(4-fluorophenyl)-2...)
Affinity DataIC50: 24nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26760(D, L mixtures | 2-fluorophenyl N-[8-(2-methyl-4,5-...)
Affinity DataIC50: 30nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26749(ethyl 8-(2-ethyl-4,5-diphenyl-1H-imidazol-1-yl)oct...)
Affinity DataIC50: 31nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26747(ethyl 6-(2-ethyl-4,5-diphenyl-1H-imidazol-1-yl)hex...)
Affinity DataIC50: 32nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26765(ethyl 7-[4,5-bis(4-fluorophenyl)-2-methyl-1H-imida...)
Affinity DataIC50: 64nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26743(ethyl 4-[4-(4,5-diphenyl-1H-imidazol-1-yl)phenoxy]...)
Affinity DataIC50: 64nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26746(ethyl 4-[3-(4,5-diphenyl-1H-imidazol-1-yl)phenoxy]...)
Affinity DataIC50: 91nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26762(D, L mixtures | 2-fluorophenyl N-[6-(2-methyl-4,5-...)
Affinity DataIC50: 110nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26750(D, L mixtures | ethyl 2-methyl-7-(2-methyl-4,5-dip...)
Affinity DataIC50: 130nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26761(2-fluorophenyl N-[2-methyl-8-(2-methyl-4,5-dipheny...)
Affinity DataIC50: 250nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26742(methyl 2-[4-(4,5-diphenyl-1H-imidazol-1-yl)phenoxy...)
Affinity DataIC50: 670nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26754(N,N-dimethyl-7-(2-methyl-4,5-diphenyl-1H-imidazol-...)
Affinity DataIC50: 970nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26753(N-methyl-7-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl...)
Affinity DataIC50: 1.70E+3nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26745(methyl 2-[3-(4,5-diphenyl-1H-imidazol-1-yl)phenoxy...)
Affinity DataIC50: 6.50E+3nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26751(D, L mixtures | ethyl 2-ethyl-7-(2-methyl-4,5-diph...)
Affinity DataIC50: 9.90E+3nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26755(3-methyl-1-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1...)
Affinity DataIC50: 1.00E+4nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26756(3-[6-(2-methyl-4,5-diphenyl-1H-imidazol-1-yl)hexyl...)
Affinity DataIC50: 1.00E+4nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26744(ethyl 5-[4-(4,5-diphenyl-1H-imidazol-1-yl)phenoxy]...)
Affinity DataIC50: 1.00E+4nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26763(2-fluorophenyl N-ethyl-N-[6-(2-methyl-4,5-diphenyl...)
Affinity DataIC50: 1.00E+5nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26764(2-fluorophenyl N-[6-(2-methyl-4,5-diphenyl-1H-imid...)
Affinity DataIC50: 1.00E+5nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Bristol-Myers Squibb

LigandPNGBDBM26752(D, L mixtures | ethyl 7-(2-methyl-4,5-diphenyl-1H-...)
Affinity DataIC50: 1.00E+5nMpH: 9.0 T: 2°CAssay Description:FAAH Inhibition Assay [3H]Ethanolamine produced from [3H]AEA hydrolysis was used to calculate FAAH activity and was measured by scintillation countin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2009
Entry Details Article
PubMed