Compile Data Set for Download or QSAR
Report error Found 110 Enz. Inhib. hit(s) with all data for entry = 50020236
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211565((R)-N-[(S)-1-(2-aminomethyl-5-chloro-benzylcarbamo...)
Affinity DataKi:  0.0330nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211578((S)-1-[(R)-4-(1-oxy-pyridin-2-yl)-2-phenylmethanes...)
Affinity DataKi:  0.0490nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211567((R)-N-[(S)-1-(2-aminomethyl-5-chloro-benzylcarbamo...)
Affinity DataKi:  0.0590nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211585([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211571((R)-N-((S)-1-(2-(aminomethyl)-5-chlorobenzylamino)...)
Affinity DataKi:  0.0840nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211564((R)-N-[(5-chloro-2-ethyl-benzylcarbamoyl)-methyl]-...)
Affinity DataKi:  0.0950nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211563((S)-4-(2-aminomethyl-5-chloro-benzylcarbamoyl)-4-{...)
Affinity DataKi:  0.240nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211570(N-((S)-1-(2-(aminomethyl)-5-chlorobenzylamino)-3-h...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211582((R)-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-4...)
Affinity DataKi:  0.320nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211552((4-{[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211572((4-{[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-...)
Affinity DataKi:  0.360nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211586((s)-4-(2-aminomethyl-5-chloro-benzylcarbamoyl)-4-[...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211578((S)-1-[(R)-4-(1-oxy-pyridin-2-yl)-2-phenylmethanes...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211587(N-[(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarb...)
Affinity DataKi:  0.630nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211584([1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-meth...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211551(N-[1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbamoy...)
Affinity DataKi:  0.870nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211576([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211556([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  0.940nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211577([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  1nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211581(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211580([1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-meth...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211566([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211555(N-[(2,5-dichloro-benzylcarbamoyl)-methyl]-4-(1-oxy...)
Affinity DataKi:  2.55nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211573(ethyl 2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobe...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211562(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211575((R)-N-[(3-chloro-benzylcarbamoyl)-methyl]-4-(1-oxy...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211560(N-[(2-aminomethyl-5-chloro-benzylcarbamoyl)-methyl...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211581(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211559(ethyl 2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobe...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211573(ethyl 2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobe...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211557(N-[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-me...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211566([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211568(N-[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-me...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211585([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211576([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  7.80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211562(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211577([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  9nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211554([1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-meth...)
Affinity DataKi:  16nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211559(ethyl 2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobe...)
Affinity DataKi:  17nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211556([(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbam...)
Affinity DataKi:  17.3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211587(N-[(R)-1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarb...)
Affinity DataKi:  17.7nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211551(N-[1-[(S)-2-(2-aminomethyl-5-chloro-benzylcarbamoy...)
Affinity DataKi:  19nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211561(N-{[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-methyl...)
Affinity DataKi:  21nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211571((R)-N-((S)-1-(2-(aminomethyl)-5-chlorobenzylamino)...)
Affinity DataKi:  24nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211553(N-[(2-aminomethyl-benzylcarbamoyl)-methyl]-4-(1-ox...)
Affinity DataKi:  32nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211569(4-(1-oxy-pyridin-2-yl)-2-phenylmethanesulfonylamin...)
Affinity DataKi:  52nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211558(N-{[(5-chloro-thiophen-2-ylmethyl)-carbamoyl]-meth...)
Affinity DataKi:  53nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211583(N-[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-me...)
Affinity DataKi:  65nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211565((R)-N-[(S)-1-(2-aminomethyl-5-chloro-benzylcarbamo...)
Affinity DataKi:  170nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211564((R)-N-[(5-chloro-2-ethyl-benzylcarbamoyl)-methyl]-...)
Affinity DataKi:  170nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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