Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50020243
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211650(3-(4-(4-((1-(2-chlorocyclopent-1-enyl)ethoxy)carbo...)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211649(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211647(3-(4-(4-((1-(2-chlorocyclohex-1-enyl)ethoxy)carbon...)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211646(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 72nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211655(4-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 73nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211645(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 74nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211651(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 81nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211648(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211653(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211654(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 120nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211648(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211650(3-(4-(4-((1-(2-chlorocyclopent-1-enyl)ethoxy)carbo...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211655(4-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211647(3-(4-(4-((1-(2-chlorocyclohex-1-enyl)ethoxy)carbon...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211646(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211649(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211651(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211653(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211654(5-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 370nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211645(2-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonyl)isoxaz...)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Rat)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211652(3-{2'-[1-(2-chloro-phenyl)-ethoxycarbonylamino]-bi...)
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at LPA1 receptor in rat hepatic stellate cells assessed as inhibition of lysophosphatidic acid-induced intracellular calcium infl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50211652(3-{2'-[1-(2-chloro-phenyl)-ethoxycarbonylamino]-bi...)
Affinity DataIC50: 4.00E+4nMAssay Description:Antagonist activity at human recombinant LPA1 receptor expressed in CHOK1 cells assessed as inhibition of lysophosphatidic acid-induced intracellular...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed