Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50020313
TargetSodium channel protein type 10 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 8nMAssay Description:Inhibition of inactivated human Nav1.8 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 3 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 2.45E+3nMAssay Description:Inhibition of inactivated human Nav1.3 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 6.74E+3nMAssay Description:Inhibition of inactivated human Nav1.7 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 7.18E+3nMAssay Description:Inhibition of inactivated human Nav1.2 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50212239(5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-...)
Affinity DataIC50: 7.44E+3nMAssay Description:Inhibition of inactivated human Nav1.5 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 10 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50178861(trans-N1-methyl-N1-((2'-sulfamoylbiphenyl-4-yl)met...)
Affinity DataKi:  180nMAssay Description:Binding affinity to Nav1.8 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50178861(trans-N1-methyl-N1-((2'-sulfamoylbiphenyl-4-yl)met...)
Affinity DataKi:  250nMAssay Description:Binding affinity to Nav1.7 sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed