Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50042259
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423011(CHEMBL267996)
Affinity DataEC50: <1.00E+4nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataEC50:  1.00E+3nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423013(CHEMBL395527)
Affinity DataEC50:  631nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423008(CHEMBL230804)
Affinity DataEC50: <1.00E+4nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423012(CHEMBL266742)
Affinity DataEC50: <1.00E+4nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50085046(2-(1-Carboxy-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-y...)
Affinity DataEC50:  0.630nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423007(CHEMBL398185)
Affinity DataEC50: <1.00E+4nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423009(CHEMBL230731)
Affinity DataEC50:  631nMAssay Description:Transactivation of human PPARgamma in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423007(CHEMBL398185)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423008(CHEMBL230804)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423013(CHEMBL395527)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423009(CHEMBL230731)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423012(CHEMBL266742)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423011(CHEMBL267996)
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50085046(2-(1-Carboxy-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of BRL-49653 stimulated human PPARgamma transactivation in CV-1 cells by GAL4 reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002865(CHEMBL230730)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002864(CHEMBL398183)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423009(CHEMBL230731)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002863(CHEMBL230732)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423013(CHEMBL395527)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002862(CHEMBL396220)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423011(CHEMBL267996)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002860(CHEMBL231656)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002868(CHEMBL230523)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423010(CHEMBL230259)
Affinity DataKi:  138nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002858(CHEMBL230524)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002859(CHEMBL396480)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002866(CHEMBL266741)
Affinity DataKi:  166nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002867(CHEMBL396481)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423012(CHEMBL266742)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002869(CHEMBL230522)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423008(CHEMBL230804)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002870(CHEMBL266985)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50002871(CHEMBL396987)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423007(CHEMBL398185)
Affinity DataKi:  912nMAssay Description:Displacement of [3H]BRL49653 from PPARgamma by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed