Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50020484
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214466(N-(3-(8-cyano-4-(cyclopropylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  0.260nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214473(N-(3-(8-CYANO-4-(PHENYLAMINO)PYRAZOLO[1,5-A][1,3,5...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214454(N-(3-(8-cyano-4-(cyclobutylamino)pyrazolo[1,5-a][1...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214444(2-(p-toluidino)-4-(phenylamino)pyrazolo[1,5-a][1,3...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214465(2-(4-chlorobenzylamino)-4-(phenylamino)pyrazolo[1,...)
Affinity DataKi:  5nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214477(4-(phenylamino)-2-(4-(pyridin-2-yl)piperazin-1-yl)...)
Affinity DataKi:  7nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214474(N-(3-(8-cyano-4-(phenethylamino)pyrazolo[1,5-a][1,...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214460(2-(CYCLOHEXYLMETHYLAMINO)-4-(PHENYLAMINO)PYRAZOLO[...)
Affinity DataKi:  8nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214448(2-(3,4-dimethoxyphenylamino)-4-(phenylamino)pyrazo...)
Affinity DataKi:  9nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214450(2-(3,4-dihydroisoquinolin-2(1H)-yl)-4-(phenylamino...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214464(N-(3-(8-methyl-4-(phenylamino)pyrazolo[1,5-a][1,3,...)
Affinity DataKi:  11nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214457(2-(2,3-dihydro-1H-inden-2-ylamino)-4-(phenylamino)...)
Affinity DataKi:  12nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214453(2-(isopentylamino)-4-(phenylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  13nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214468(4-(phenylamino)-2-(pyrrolidin-1-yl)pyrazolo[1,5-a]...)
Affinity DataKi:  14nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214446(2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine...)
Affinity DataKi:  15nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214443(N-(3-(8-bromo-4-(cyclopropylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  17nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214471(2-(4-(diethylamino)phenylamino)-4-(phenylamino)pyr...)
Affinity DataKi:  23nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214446(2,4-bis(phenylamino)pyrazolo[1,5-a][1,3,5]triazine...)
Affinity DataKi:  24nMAssay Description:Inhibition of corn CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214452(2-(4-ETHYLPIPERAZIN-1-YL)-4-(PHENYLAMINO)PYRAZOLO[...)
Affinity DataKi:  24nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214451(N-(3-(4-(cyclopropylamino)-8-methylpyrazolo[1,5-a]...)
Affinity DataKi:  35nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214470(2-(1H-imidazol-2-ylamino)-4-(phenylamino)pyrazolo[...)
Affinity DataKi:  45nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214478(2-(benzyl(methyl)amino)-4-(phenylamino)pyrazolo[1,...)
Affinity DataKi:  55nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214445(3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-...)
Affinity DataKi:  95nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214479(2-(1H-imidazol-1-yl)-4-(phenylamino)pyrazolo[1,5-a...)
Affinity DataKi:  126nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214456(2-(p-toluidino)-4-(phenethylamino)pyrazolo[1,5-a][...)
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214475(4-(2-(1H-IMIDAZOL-4-YL)ETHYLAMINO)-2-(PHENYLAMINO)...)
Affinity DataKi:  137nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214459(4-(phenylamino)-2-(pyridin-3-ylamino)pyrazolo[1,5-...)
Affinity DataKi:  168nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214462(N-(3-(8-cyano-4-(3-ethoxyphenylamino)pyrazolo[1,5-...)
Affinity DataKi:  190nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214449(N-(3-(8-cyano-4-(3-(difluoromethoxy)phenylamino)py...)
Affinity DataKi:  190nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214461(3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-...)
Affinity DataKi:  190nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214455(N-(3-(8-cyano-4-(4-(piperazin-1-ylmethyl)phenylami...)
Affinity DataKi:  210nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214458(2-(methyl(phenyl)amino)-4-(phenylamino)pyrazolo[1,...)
Affinity DataKi:  242nMAssay Description:Inhibition of corn CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Maize)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214472(N2,N4-diphenylpyrazolo[1,5-a][1,3,5]triazine-2,4-d...)
Affinity DataKi:  260nMAssay Description:Inhibition of corn CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214447(3-(2-(3-acetamidophenylamino)-8-cyanopyrazolo[1,5-...)
Affinity DataKi:  370nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214469(N-(3-(8-cyano-4-(4-((diethylamino)methyl)phenylami...)
Affinity DataKi:  500nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214463(N-(3-(8-cyano-4-(3-(diethylamino)phenylamino)pyraz...)
Affinity DataKi:  550nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214442(N-(3-(8-cyano-4-(3-(pyrrolidine-1-carbonyl)phenyla...)
Affinity DataKi:  700nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214476(N-(3-(4-(cyclopropylamino)-8-ethylpyrazolo[1,5-a][...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha(Human)
Polaris Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50214467(4-(phenethylamino)-2-(pyridin-3-ylamino)pyrazolo[1...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human CK2 alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed