Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50020553
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human SST5 receptor expressed in CHOK1 cells assessed as effect on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 1.20nMAssay Description:Agonist activity at human SST5 receptor expressed in CHOK1 cells assessed as effect on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50: 73nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: 75nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 83nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50: 89nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50: 103nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexah...)
Affinity DataIC50: 129nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST4 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 233nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: 245nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataIC50: 251nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexah...)
Affinity DataIC50: 318nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexah...)
Affinity DataIC50: 357nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215026((2S)-6-amino-N-benzyl-2-[(4R)-4-[(3,3-diphenylprop...)
Affinity DataIC50: 694nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexah...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215027(5-[(4R)-3-oxo-4-[(phenylacetyl)amino]-3,4,5,10-tet...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50215028(N-[(4R)-2-(5-aminopentyl)-3-oxo-1,2,3,4,5,10-hexah...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I][Leu8-D-Trp22, Tyr25]-SRIF28 from human SST1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed