Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50021079
LigandPNGBDBM50220714(N-((1s,4s)-4-hydroxy-4-(5-hydroxypyridin-2-yl)cycl...)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220726(N-((1s,4s)-4-(3-fluoro-4-hydroxyphenyl)-4-hydroxyc...)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220729(N-((1s,4s)-4-hydroxy-4-(4-hydroxyphenyl)cyclohexyl...)
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220712(N-((1s,4s)-4-hydroxy-4-(4-hydroxy-2-methylphenyl)c...)
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220716(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-phenyl...)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220727(N-((1r,4r)-4-(3-fluoro-4-hydroxyphenyl)cyclohexyl)...)
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220720(N-((1s,4s)-4-hydroxy-4-(2-oxo-2,3-dihydrooxazolo[4...)
Affinity DataIC50: 85nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220725(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(5-met...)
Affinity DataIC50: 96nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220728(N-((1s,4s)-4-hydroxy-4-(5-hydroxy-4-methylpyridin-...)
Affinity DataIC50: 116nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220715(N-((1s,4s)-4-hydroxy-4-(4-hydroxy-3-methylphenyl)c...)
Affinity DataIC50: 189nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220713(N-((1r,4r)-4-(4-hydroxy-2-methylphenyl)cyclohexyl)...)
Affinity DataIC50: 722nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220718(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(pyrid...)
Affinity DataIC50: 856nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220734(2-(dimethylamino)-N-((1r,4r)-4-(4-hydroxyphenyl)cy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220723(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-1,2,3,4-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220731(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(1-met...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220719(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(pyrid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220730((R)-6-(2-(4-(3-fluorophenyl)-4-hydroxypiperidin-1-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220732(N-((1s,4s)-4-hydroxy-4-(1H-pyrazol-4-yl)cyclohexyl...)
Affinity DataIC50: 2.44E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220735(N-((1s,4s)-4-(1H-benzo[d]imidazol-5-yl)-4-hydroxyc...)
Affinity DataIC50: 4.96E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220724(N-((1s,4s)-4-hydroxy-4-(6-(methylsulfonamido)pyrid...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220722(N-((1r,4r)-4-(4-hydroxy-3-methylphenyl)cyclohexyl)...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220721(N-((1s,4s)-4-hydroxy-4-(1H-imidazol-4-yl)cyclohexy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220717(N-((1s,4s)-4-(6-aminopyridin-3-yl)-4-hydroxycycloh...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]CP-101606 from NR2B in rat forebrain P2 membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220725(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(5-met...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220726(N-((1s,4s)-4-(3-fluoro-4-hydroxyphenyl)-4-hydroxyc...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220723(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-1,2,3,4-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220733(4-benzyl-1-(2-hydroxy-2-(4-hydroxyphenyl)ethyl)pip...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220719(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(pyrid...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220718(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-(pyrid...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220714(N-((1s,4s)-4-hydroxy-4-(5-hydroxypyridin-2-yl)cycl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220729(N-((1s,4s)-4-hydroxy-4-(4-hydroxyphenyl)cyclohexyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220716(N-((1r,4r)-4-(4-hydroxyphenyl)cyclohexyl)-3-phenyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50220713(N-((1r,4r)-4-(4-hydroxy-2-methylphenyl)cyclohexyl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of [3H]dofetilide from human HERG expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed