Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50021205
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in mouse LV2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222059(N-[3-chloro-4-(3-oxo-2,3-dihydro-1H,5H-benzo[e]pyr...)
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222058(N-[3-chloro-4-(3-oxo-11,11a-dihydro-3H,5H-benzo[e]...)
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177593((5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)...)
Affinity DataIC50: 80.3nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in mouse LV2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 124nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177593((5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)...)
Affinity DataIC50: 353nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065115(N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][1,4]diazepine-...)
Affinity DataIC50: 519nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50177593((5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)...)
Affinity DataIC50: 778nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222060(1-(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benza...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222060(1-(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benza...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222059(N-[3-chloro-4-(3-oxo-2,3-dihydro-1H,5H-benzo[e]pyr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222060(1-(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benza...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222059(N-[3-chloro-4-(3-oxo-2,3-dihydro-1H,5H-benzo[e]pyr...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222057(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222057(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222057(2-(2-chloro-4-(5-fluoro-2-methylbenzamido)benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222058(N-[3-chloro-4-(3-oxo-11,11a-dihydro-3H,5H-benzo[e]...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]oxytocin from human oxytocin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222058(N-[3-chloro-4-(3-oxo-11,11a-dihydro-3H,5H-benzo[e]...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]manning ligand from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50222061(10-[2-chloro-4-(3-methyl-pyrazol-1-yl)-benzoyl]-1,...)
Affinity DataIC50: 1.21E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in mouse LV2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed