Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50003894
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  0.643nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(Biriperone | 1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(Biriperone | 1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477151(CHEMBL393622)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477151(CHEMBL393622)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(Biriperone | 1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a...)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  2.25E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477150(CHEMBL240733)
Affinity DataKi: <1.00E+5nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477150(CHEMBL240733)
Affinity DataKi: <1.00E+5nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed