Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50021552
TargetMAP kinase-activated protein kinase 2(Human)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50225787(CHEMBL397819 | CHEMBL1185204 | 2,4-diamino-6,7-dih...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MK2 in human TERT immortalised HCA2 cells assessed as inhibition of anisomycin-induced HSP27 phosphorylation by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Cardiff University

Curated by ChEMBL
LigandPNGBDBM50411445(CHEMBL235658)
Affinity DataKi:  330nMAssay Description:Inhibition of MK2 in human TERT immortalised HCA2 cells assessed as inhibition of anisomycin-induced HSP27 phosphorylation at 2.5 uM by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed