Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50038267
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50266539(CHEMBL456066 | (4S,4aS,5aS,6S,12aS)-7-chloro-4-(di...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50422012(Klinomycin | Minocin | Vectrin | MINOCYCLINE)
Affinity DataIC50: 6.20E+5nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50368781(Achromycin | Cyclopar | Liquamycin | Panmycin | TE...)
Affinity DataIC50: 7.80E+5nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM52947(cid_16746590 | Doxycycline hyclate | (2Z,4S,4aR,5S...)
Affinity DataIC50: 8.60E+5nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50423606(Chlorodeoxylincomycin | Chlorolincomycin | U-21251...)
Affinity DataIC50: 5.10E+6nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50029770(4-amino-N-(5-methyl-isoxazol-3-yl)-benzenesulfonam...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM60918(5-Amino-2-hydroxy-benzoic acid | cid_4075 | MLS001...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50373919(Azasan | AZATHIOPRINE)
Affinity DataIC50: 8.10E+6nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50373918(Azasite | AZITHROMYCIN | US20240118263, Compound A...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50054601(5-methyl-N-[4-(trifluoromethyl)phenyl]-1,2-oxazole...)
Affinity DataIC50: 2.40E+6nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM18050(MTX | cid_126941 | Methotrexate | 2-[(4-{[(2,4-dia...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50366387(STREPTOMYCIN)
Affinity DataIC50: 1.80E+6nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM39340(MLS000069725 | cid_5336 | SMR000058213 | SULFAPYRI...)
Affinity DataIC50: 1.00E+7nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM18069(CHEMBL22 | TMP | Trimethoprim (TMP) | 5-[(3,4,5-tr...)
Affinity DataIC50: 7.50E+6nMAssay Description:Inhibition of PAD4 by ABPP-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50266539(CHEMBL456066 | (4S,4aS,5aS,6S,12aS)-7-chloro-4-(di...)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition of PAD4 measured by intercept plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50422012(Klinomycin | Minocin | Vectrin | MINOCYCLINE)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition of PAD4 measured by intercept plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50422012(Klinomycin | Minocin | Vectrin | MINOCYCLINE)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of PAD4 measured by slope plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50266539(CHEMBL456066 | (4S,4aS,5aS,6S,12aS)-7-chloro-4-(di...)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of PAD4 measured by slope plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50366387(STREPTOMYCIN)
Affinity DataKi:  5.60E+5nMAssay Description:Inhibition of PAD4 measured by slope plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
TargetProtein-arginine deiminase type-4(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM52947(cid_16746590 | Doxycycline hyclate | (2Z,4S,4aR,5S...)
Affinity DataKi:  6.30E+5nMAssay Description:Inhibition of PAD4 measured by intercept plot of Lineweaver-Burke analysesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed