Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50025605
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 130nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247392(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 150nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 150nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 150nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 160nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 170nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247396(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 260nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247417(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 280nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 300nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 450nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247431(N-Benzyl-8-isopopyl-9-oxo-8,9-dihydro[1,3]thiazolo...)
Affinity DataIC50: 520nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186073(N-(2-Dimethylamino-ethyl)-8-isopopyl-9-oxo-8,9-dih...)
Affinity DataIC50: 560nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247391(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 640nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186084(N-(2-Dimethylamino-ethyl)-8-ethyl-9-oxo-8,9-dihydr...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247392(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247419(N-Benzyl-8-ethyl-9-oxo-8,9-dihydrothiazolo[5,4-f]q...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247417(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186073(N-(2-Dimethylamino-ethyl)-8-isopopyl-9-oxo-8,9-dih...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247394(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247391(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247396(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186082(N-Isopropyl-8-ethyl-9-oxo-8,9-dihydrothiazolo[5,4-...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247431(N-Benzyl-8-isopopyl-9-oxo-8,9-dihydro[1,3]thiazolo...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247431(N-Benzyl-8-isopopyl-9-oxo-8,9-dihydro[1,3]thiazolo...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186072(N,8-diisopropyl-9-oxo-8,9-dihydrothiazolo[5,4-f]qu...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186073(N-(2-Dimethylamino-ethyl)-8-isopopyl-9-oxo-8,9-dih...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247419(N-Benzyl-8-ethyl-9-oxo-8,9-dihydrothiazolo[5,4-f]q...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186073(N-(2-Dimethylamino-ethyl)-8-isopopyl-9-oxo-8,9-dih...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186084(N-(2-Dimethylamino-ethyl)-8-ethyl-9-oxo-8,9-dihydr...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247395(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247372(8-Ethyl-9-oxo-8,9-dihydro-6-thiazolo[5,4-f]quinazo...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CDK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186082(N-Isopropyl-8-ethyl-9-oxo-8,9-dihydrothiazolo[5,4-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247431(N-Benzyl-8-isopopyl-9-oxo-8,9-dihydro[1,3]thiazolo...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247419(N-Benzyl-8-ethyl-9-oxo-8,9-dihydrothiazolo[5,4-f]q...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50186072(N,8-diisopropyl-9-oxo-8,9-dihydrothiazolo[5,4-f]qu...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK1/cyclinBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247393(8-Ethyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quinazoli...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Université

Curated by ChEMBL
LigandPNGBDBM50247418(8-Isopropyl-9-oxo-8,9-dihydro-thiazolo[5,4-f]quina...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CDK5/p25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Université

Curated by ChEMBL
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of GSK3alpha/betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed