Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50021647
LigandPNGBDBM50226429([L-arginyl]-N-(2,4-dichlorophenethyl)glycine 2,4-(...)
Affinity DataIC50: 170nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226436([L-arginyl]-[N-(2,4-dichlorophenethyl)glycyl]-N-[2...)
Affinity DataIC50: 180nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226431([[N-(2,4-dichlorophenethyl)-N-(6-aminohexyl)]glycy...)
Affinity DataIC50: 400nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226430([L-arginyl]-[N-[2-(indol-3-yl)ethyl]glycyl]-N-(2,4...)
Affinity DataIC50: 520nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226432(cis-(L-arginyl)amino-N-(2,4-dichlorophenylmethyl)-...)
Affinity DataIC50: 700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226435((S)-N-(2,4-dichlorophenethyl)-N-(2-((2,4-dichlorop...)
Affinity DataIC50: 700nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226429([L-arginyl]-N-(2,4-dichlorophenethyl)glycine 2,4-(...)
Affinity DataIC50: 800nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226434([L-arginyl]-N-[2-(indol-3-yl)ethyl]glycine 2-(indo...)
Affinity DataIC50: 1.10E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50226433([L-arginyl]-[N-[2-(indol-3-yl)-ethyl]glycyl]-N-[(2...)
Affinity DataIC50: 1.33E+3nMAssay Description:Blockade of capsaicin-activated rat TRPV1 channel expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226431([[N-(2,4-dichlorophenethyl)-N-(6-aminohexyl)]glycy...)
Affinity DataIC50: 3.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226432(cis-(L-arginyl)amino-N-(2,4-dichlorophenylmethyl)-...)
Affinity DataIC50: 8.00E+3nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226435((S)-N-(2,4-dichlorophenethyl)-N-(2-((2,4-dichlorop...)
Affinity DataIC50: 1.50E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226430([L-arginyl]-[N-[2-(indol-3-yl)ethyl]glycyl]-N-(2,4...)
Affinity DataIC50: 1.70E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226434([L-arginyl]-N-[2-(indol-3-yl)ethyl]glycine 2-(indo...)
Affinity DataIC50: 1.80E+4nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226436([L-arginyl]-[N-(2,4-dichlorophenethyl)glycyl]-N-[2...)
Affinity DataIC50: 1.66E+5nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rat)
University of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226433([L-arginyl]-[N-[2-(indol-3-yl)-ethyl]glycyl]-N-[(2...)
Affinity DataIC50: 2.07E+5nMAssay Description:Blockade of L-glutamate/glycine-activated rat NR1/NR2A NMDA receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed